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MSc theses (1)
Andrej Emanuel Cotman:
Načrtovanje in sinteza analogov 4,5-dibromo-1H-pirola s tirozinskim fragmentom kot zaviralcev giraze B s protibakterijskim delovanjem
Other documents (16)
Martina Durcik, Andrej Emanuel Cotman, Žan Toplak, Štefan Možina, Žiga Skok, Maria Vittoria Piras, Nace Zidar, Janez Ilaš, Anamarija Zega, Jurij Trontelj, Danijel Kikelj, Tihomir Tomašič, Lucija Peterlin-Mašič:
New dual inhibitors of bacterial topoisomerases with broad-spectrum antibacterial activity and in vivo efficacy against vancomycin-intermediate Staphylococcus aureus
Jaka Dernovšek, Živa Zajec, Dunja Urbančič, Irena Mlinarič-Raščan, Andrej Emanuel Cotman, Nace Zidar, Tihomir Tomašič:
Exploration and optimisation of structure-activity relationships of new triazole-based C-terminal Hsp90 inhibitors towards in vivo anticancer potency
Miha Virant, Mateja Mihelač, Martin Gazvoda, Andrej Emanuel Cotman, Anja Frantar, Balazs Pinter, Janez Košmrlj:
Pyridine wingtip in ▫$[Pd(Py-tzNHC)_2]^{2+}$▫ complex is a proton shuttle in the catalytic hydroamination of alkynes
Nace Zidar, Alessia Onali, Peter Peršolja, Davide Benedetto Tiz, Jaka Dernovšek, Žiga Skok, Martina Durcik, Andrej Emanuel Cotman, Martina Hrast Rambaher, Anamarija Zega, Lucija Peterlin-Mašič, Janez Ilaš, Tihomir Tomašič, Danijel Kikelj:
Improved N-phenylpyrrolamide inhibitors of DNA gyrase as antibacterial agents for high-priority bacterial strains
Andrej Emanuel Cotman, Pavel A. Dub, Maša Sterle, Matic Lozinšek, Jaka Dernovšek, Živa Zajec, Anamarija Zega, Tihomir Tomašič, Dominique Cahard:
Catalytic stereoconvergent synthesis of homochiral β‑CF$_3$, β‑SCF$_3$, and β‑OCF$_3$ benzylic alcohols
Andrej Emanuel Cotman, Martina Durcik, Davide Benedetto Tiz, Federica Fulgheri, Daniela Secci, Maša Sterle, Štefan Možina, Žiga Skok, Nace Zidar, Anamarija Zega, Janez Ilaš, Lucija Peterlin-Mašič, Tihomir Tomašič, Danijel Kikelj:
Discovery and hit-to-lead optimization of benzothiazole scaffold-based DNA gyrase inhibitors with potent activity against Acinetobacter baumannii and Pseudomonas aeruginosa
Maša Sterle, Matej Huš, Matic Lozinšek, Anamarija Zega, Andrej Emanuel Cotman:
Hydrogen-bonding ability of Noyori–Ikariya catalysts enables stereoselective access to CF$_3$-substituted syn-1,2-diols via dynamic kinetic resolution
Maša Sterle, Martina Durcik, Danijel Kikelj, Nace Zidar, Lucija Peterlin-Mašič, Janez Ilaš, Tihomir Tomašič, Andrej Emanuel Cotman, Anamarija Zega:
Exploring the 5-substituted 2-aminobenzothiazole-based DNA gyrase B inhibitors active against ESKAPE pathogens
Simona Hašanová, Jernej Cingl, Tihomir Tomašič, Andrej Emanuel Cotman:
Catalytic performance of Noyori–Ikariya-type ruthenium complex with tethered syn-ULTAM ligand for the asymmetric transfer hydrogenation of ketones
Nace Zidar, Andrej Emanuel Cotman, Wessel Sinnige, Ondřej Benek, Michaela Barančokova, Anamarija Zega, Lucija Peterlin-Mašič, Tihomir Tomašič, Janez Ilaš, Ricardo D. Enriz, Danijel Kikelj:
Exploring the interaction of N-(benzothiazol-2-yl)pyrrolamide DNA gyrase inhibitors with the GyrB ATP-binding site lipophilic floor
Andrej Emanuel Cotman, Federica Fulgheri, Martina Piga, Peter Peršolja, Davide Benedetto Tiz, Žiga Skok, Martina Durcik, Maša Sterle, Jaka Dernovšek, Anamarija Zega, Lucija Peterlin-Mašič, Janez Ilaš, Tihomir Tomašič, Danijel Kikelj, Nace Zidar:
New N-phenylpyrrolamide inhibitors of DNA gyrase with improved antibacterial activity
Maša Zorman, Maja Kokot, Irena Zdovc, Lidija Šenerović, Mina Mandic, Nace Zidar, Andrej Emanuel Cotman, Martina Durcik, Lucija Peterlin-Mašič, Nikola Minovski, Marko Anderluh, Martina Hrast Rambaher:
Enhancing antibacterial efficacy
Ivan Džajić, Tihomir Tomašič, Luis Pardo A., Lucija Peterlin-Mašič, Andrej Emanuel Cotman:
Lipophilic cations as mitochondria-targeting moieties
Ivan Džajić:
Načrtovanje, sinteza in vrednotenje kvarternih dušikovih heterociklov kot fragmentov za ciljanje mitohondrijev
Ivan Džajić, Natalija Trunkelj, Jernej Repas, Maša Kandušer, Lara Smrdel, Stane Pajk, Lovro Žiberna, Irena Mlinarič-Raščan, Boštjan Markelc, Maša Omerzel, Tanja Jesenko, Tihomir Tomašič, Lucija Peterlin-Mašič, Andrej Emanuel Cotman:
Mitochondria-targeting moieties based on N-tethered pyridinium cations
Boštjan Adamlje, Tihomir Tomašič, Christian Steinebach, Sebastian Ebeling, Alexander Herrmann, Marcus D. Hartmann, Jessica L. Horner, Kinjal Bhadresha, Izidor Sosič, Andrej Emanuel Cotman:
Fluorinated aminopiperidones as non-glutarimide thalidomide analogs