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PhD theses (1)
Rok Frlan:
Načrtovanje, sinteza in vrednotenje sulfonohidrazidnih inhibitorjev Mur ligaz
MSc theses (12)
Marko Trampuž:
Načrtovanje in sinteza aminokislinskih derivatov substituiranih pirolamidov kot zaviralcev bakterijske DNA giraze B
Slavka Majcen:
Sinteza aminopirimidintiazolov s potencialnim delovanjem na napetostno odvisne ionske kanalčke
Kristina Nemec:
Sinteza derivatov 4-amino-1H-pirol-2-karboksamida s potencialnim zaviralnim delovanjem na girazo B
Andreja Jernej:
Načrtovanje in sinteza potencialnih zaviralcev giraze B z aminoetanolnim fragmentom
Andrej Emanuel Cotman:
Načrtovanje in sinteza analogov 4,5-dibromo-1H-pirola s tirozinskim fragmentom kot zaviralcev giraze B s protibakterijskim delovanjem
Eva Šimunović:
Sinteza derivatov 2,4-dihidroksibenzojske kisline kot potencialnih zaviralcev ligaze D-ala-D-ala
Eva Jerič:
Načrtovanje in sinteza derivatov 3-amino-2-tioksitiazoldin-4-ona in 1H-pirol-3-amina kot potencialnih zaviralcev giraze B
Larisa Vidmar:
Sinteza derivatov 2-(2-karbamoil-5-hidroksefenoksi)ocetne kisline z zaviralnim delovanjem na encim ligazo S-Ala
Eva Shannon Schiffrer:
Načrtovanje in sinteza derivatov pirolo[1,2-a]pirazin-1(2H)-ona s potencialnim zaviralnim delovanjem na girazo B
Manca Glavan:
Načrtovanje in sinteza aminokislinskih derivatov pirol-2-karboksamida s potencialnim zaviralnim delovanjem na girazo B
Samo Kuzmič:
Načrtovanje, sinteza in vrednotenje mimetikov D-Ala-D-Ala z azidinskim gradnikom
Urška Češarek:
Razvoj sintezne metode za pripravo aminokislinskih derivatov monobaktamov
BSc theses (7)
Katarina Škof:
Selektivna sinteza amfifilnih derivatov dihidroksibenzojske kisline in dihidrosibenzaldehida z antioksidativnim delovanjem
Sonja Jus:
Novi levcinhidrazidni inhibitorji ligaz Mur
Jerneja Tanšek:
Novi treoninhidrazidni inhibitorji ligaz Mur
Vanja Stanonik:
Sinteza 3-aminobenzensulfoniltreoninskih inhibitorjev ligaz Mur
Brigita Kure:
Sinteza substituiranih malonilaminouridinskih inhibitorjev ligaz Mur
Matic Mikec:
Sinteza dihidroksibenzamidnih zaviralcev biosinteze peptidoglikana
Nina Cirkvenčič:
Načrtovanje in sinteza 2-amino-2-oksoetil-N-(arilsulfonil)karbamatov kot inhibitorjev Murc in MurD
Other documents (14)
Macarena Funes Chabán, Martina Hrast Rambaher, Rok Frlan, Dafni G. Graikioti, Constantinos M. Athanassopoulos, María Cecilia Carpinella:
Inhibition of MurA enzyme from Escherichia coli and Staphylococcus aureus by diterpenes from Lepechinia meyenii and their synthetic analogs
Martina Hrast Rambaher, Nina Gradišek, Rok Frlan, Izidor Sosič, Aljoša Bolje, Jakob Kljun, Martin Juhás, Stanislav Gobec, Stane Pajk:
Development and evaluation of novel InhA inhibitors inspired by thiadiazole and tetrahydropyran series of inhibitors
Rok Frlan, Martina Hrast Rambaher, Stanislav Gobec:
Application of the N-dibenzyl protective group in the preparation of β-lactam pseudopeptides
Matic Proj, Krištof Bozovičar, Martina Hrast Rambaher, Rok Frlan, Stanislav Gobec:
DNA-encoded library screening on two validated enzymes of the peptidoglycan biosynthetic pathway
Samo Kuzmič, Martina Hrast Rambaher, Rok Frlan:
The synthesis of (2R)-aziridine-2-carboxylic acid containing dipeptides
Matic Proj, Martina Hrast Rambaher, Gregor Bajc, Rok Frlan, Anže Meden, Matej Butala, Stanislav Gobec:
Discovery of a fragment hit compound targeting D-Ala:D-Ala ligase of bacterial peptidoglycan biosynthesis
Matic Proj, Martina Hrast Rambaher, Damijan Knez, Krištof Bozovičar, Katarina Grabrijan, Anže Meden, Stanislav Gobec, Rok Frlan:
Fragment-sized thiazoles in fragment-based drug discovery campaigns
Martina Hrast Rambaher, Irena Zdovc, Nina Kočevar Glavač, Stanislav Gobec, Rok Frlan:
Mur ligase F as a new target for the flavonoids quercitrin, myricetin, and (–)-epicatechin
Rok Frlan, Martina Hrast Rambaher, Stanislav Gobec:
Inhibition of MurA enzyme from Escherichia coli by flavonoids and their synthetic analogues
Martina Piga, Zoltán Varga, Ádám Fehér, Ferenc Papp, Eva Korpos Pintye-Gyuri, Kavya C. Bangera, Rok Frlan, Janez Ilaš, Jaka Dernovšek, Tihomir Tomašič, Nace Zidar:
Identification of a novel structural class of H$_v$1 inhibitors by structure-based virtual screening
Tjaša Žagar, Rok Frlan, Nina Kočevar Glavač:
Using subcritical water to obtain polyphenol-rich extracts with antimicrobial properties
Damijan Knez, Fen Wang, Wen-Xiang Duan, Martina Hrast Rambaher, Stanislav Gobec, Xiao-Yu Cheng, Xiao-Bo Wang, Cheng-Jie Mao, Chun-Feng Liu, Rok Frlan:
Development of novel aza-stilbenes as a new class of selective MAO-B inhibitors for the treatment of Parkinson’s disease
Vid Kuralt, Rok Frlan:
Navigating the chemical space of ENR Inhibitors
Rok Frlan:
In silico druggability assessment of Escherichia coli FtsQ reveals tractable PPI interfaces in the divisome