271. Synthesis, biological evaluation and docking studies of benzoxazoles derived from thymoquinoneUna Glamočlija, Subhash Padhye, Selma Špirtović-Halilović, Amar Osmanović, Elma Veljović, Sunčica Roca, Irena Novaković, Boris Mandić, Iztok Turel, Jakob Kljun, Snežana Trifunović, Emira Kahrović, Sandra Kraljević-Pavelić, Anja Harej, Marko Klobučar, Davorka Završnik, 2018, izvirni znanstveni članek Ključne besede: thymoquinone, benzoxazoles, anticancer activity, antimicrobial activity, western blotting, molecular docking Celotno besedilo (datoteka, 2,92 MB) Gradivo ima več datotek! Več... |
272. Copper(II) and zinc(II) complexes with the clinically used fluconazoleNevena Lj. Stevanović, Ivana Aleksić, Jakob Kljun, Sanja Skaro-Bogojevic, Aleksandar Veselinovic, Jasmina Nikodinović-Runić, Iztok Turel, Miloš I. Djuran, Biljana Glišić, 2021, izvirni znanstveni članek Ključne besede: copper(II) complex, zinc(II) complex, fluconazole, antifungal agents, anti-biofilm activity Celotno besedilo (datoteka, 2,52 MB) Gradivo ima več datotek! Več... |
273. Structural and functional characterization of an organometallic ruthenium complex as a potential myorelaxant drugTomaž Trobec, Monika C. Žužek, Kristina Sepčić, Jerneja Kladnik, Jakob Kljun, Iztok Turel, Evelyne Benoit, Robert Frangež, 2020, izvirni znanstveni članek Ključne besede: organoruthenium nitrophenanthroline complex, acetylcholinesterase, butyrylcholinesterase, glutathione S-transferase, mouse neuromuscular system, ruthenium, muscle relaxation, physiology, glutathione transferase Celotno besedilo (datoteka, 1,45 MB) Gradivo ima več datotek! Več... |
274. Comparison of solution chemical properties and biological activity of ruthenium complexes of selected ß-diketone, 8-hydroxyquinoline and pyrithione ligandsTamás Pivarcsik, Gábor Tóth, Nikoletta Szemerédi, Anita Bogdanov, Gabriella Spengler, Jakob Kljun, Jerneja Kladnik, Iztok Turel, Éva A. Enyedy, 2021, izvirni znanstveni članek Ključne besede: MTT assay, UV-vis, solution stability, MRSA, albumin binding, ligand effect Celotno besedilo (datoteka, 5,33 MB) Gradivo ima več datotek! Več... |
275. Organoruthenium complexes with benzo-fused pyrithiones overcome platinum resistance in ovarian cancer cellsJerneja Kladnik, James P. C. Coverdale, Jakob Kljun, Hilke Burmeister, Petra Lippman, Francesca G. Ellis, Alan M. Jones, Ingo Ott, Isolda Romero-Canelón, Iztok Turel, 2021, izvirni znanstveni članek Ključne besede: ruthenium, pyrithione, resistance to chemotherapy, cancer, ovarian, thioredoxin Celotno besedilo (datoteka, 3,10 MB) Gradivo ima več datotek! Več... |
276. Tailoring copper(II) complexes with pyridine-4,5-dicarboxylate esters for anti-Candida activityTina P. Andrejević, Ivana Aleksić, Marta Počkaj, Jakob Kljun, Dušan Milivojević, Nevena Lj. Stevanović, Jasmina Nikodinović-Runić, Iztok Turel, Miloš I. Djuran, Biljana Glišić, 2021, izvirni znanstveni članek Ključne besede: copper(II) complexes, pyridine-4, 5-dicarboxylates, antimicrobial activity, Candida albicans, filamentation, DNA/BSA interaction Celotno besedilo (datoteka, 2,06 MB) Gradivo ima več datotek! Več... |
277. Clinically used antifungal azoles as ligands for gold(III) complexesNevena Lj. Stevanović, Jakob Kljun, Ivana Aleksić, Sanja Skaro-Bogojevic, Dušan Milivojević, Aleksandar Veselinovic, Iztok Turel, Miloš I. Djuran, Jasmina Nikodinović-Runić, Biljana Glišić, 2022, izvirni znanstveni članek Celotno besedilo (datoteka, 1,32 MB) Gradivo ima več datotek! Več... |
278. Ruthenium complexes show potent inhibition of AKR1C1, AKR1C2, and AKR1C3 enzymes and anti-proliferative action against chemoresistant ovarian cancer cell lineJakob Kljun, Renata Pavlič, Eva Hafner, Tanja Lipec, Sara Moreno-Da Silva, Primož Tič, Iztok Turel, Tomaž Büdefeld, Jure Stojan, Tea Lanišnik-Rižner, 2022, izvirni znanstveni članek Ključne besede: ruthenium complexes, synthesis, crystal structure, anticancer, aldo-keto reductase, enzyme inhibition Celotno besedilo (datoteka, 1,85 MB) Gradivo ima več datotek! Več... |
279. Zinc pyrithione is a potent inhibitor of PL$^{Pro}$ and cathepsin L enzymes with ex vivo inhibition of SARS-CoV-2 entry and replicationJerneja Kladnik, Ana Dolinar, Jakob Kljun, David Perea, Judith Grau-Expósito, Meritxell Genescà, Marko Novinec, Maria J. Buzon, Iztok Turel, 2022, izvirni znanstveni članek Ključne besede: antiviral agents, SARS-CoV-2, inhibition, pyrithione, zinc Celotno besedilo (datoteka, 1,91 MB) Gradivo ima več datotek! Več... |
280. Silver(I) complexes with voriconazole as promising anti-Candida agentsMia Stanković, Sanja Skaro-Bogojevic, Jakob Kljun, Žiko Milanović, Nevena Lj. Stevanović, Jelena Lazić, Sandra Vojnović, Iztok Turel, Miloš I. Djuran, Biljana Glišić, 2024, izvirni znanstveni članek Ključne besede: silver(I) complexes, Voriconazole, coordination polymers, DFT calculations, anti-Candida activity, CYP51B Celotno besedilo (datoteka, 4,80 MB) Gradivo ima več datotek! Več... |