21. Amide containing NBTI antibacterials with reduced hERG inhibition, retained antimicrobial activity against gram-positive bacteria and in vivo efficacyMaja Kokot, Matjaž Weiss, Irena Zdovc, Lidija Senerovic, Natasa Radakovic, Marko Anderluh, Nikola Minovski, Martina Hrast, 2023, izvirni znanstveni članek Ključne besede: NBTIs, DNA gyrase, topoisomerase IV, antibacterials, MRSA, hERG inhibition, in vivo efficacy Celotno besedilo (datoteka, 3,61 MB) Gradivo ima več datotek! Več... |
22. Intracellular hydrolysis of small-molecule O-linked N-acetylglucosamine transferase inhibitors differs among cells and is not required for its inhibitionElena Maria Loi, Matjaž Weiss, Stane Pajk, Martina Gobec, Tihomir Tomašič, Roland J. Pieters, Marko Anderluh, 2020, izvirni znanstveni članek Ključne besede: ester hydrolysis, inhibitor, O-GlcNAc transferase, OGT inhibitor Celotno besedilo (datoteka, 1,90 MB) Gradivo ima več datotek! Več... |
23. Inhibition of O-GlcNAc transferase alters the differentiation and maturation process of human monocyte derived dendritic cellsMatjaž Weiss, Marko Anderluh, Martina Gobec, 2021, izvirni znanstveni članek Ključne besede: O-GlcNAcylation, O-GlcNAc transferase (OGT), monocyte derived DCs, OSMI-1, immunometabolism, pharmaceutical chemistry Celotno besedilo (datoteka, 2,84 MB) Gradivo ima več datotek! Več... |
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25. Structurally optimized potent dual-targeting NBTI antibacterials with an enhanced bifurcated halogen-bonding propensityMaja Kokot, Matjaž Weiss, Irena Zdovc, Martina Hrast, Marko Anderluh, Nikola Minovski, 2021, izvirni znanstveni članek Ključne besede: NBTIs, DNA gyrase, topoisomerase IV, bifurcated halogen bonds, dual targeting Celotno besedilo (datoteka, 2,92 MB) Gradivo ima več datotek! Več... |
26. New quinolinone O-GlcNAc transferase inhibitors based on fragment growthMatjaž Weiss, Elena Maria Loi, Maša Sterle, Cyril Balsollier, Tihomir Tomašič, Roland J. Pieters, Martina Gobec, Marko Anderluh, 2021, izvirni znanstveni članek Ključne besede: O-GlcNAc, O-GlcNAc transferase, protein glycosylation, fragments growth, molecular docking Celotno besedilo (datoteka, 1,37 MB) Gradivo ima več datotek! Več... |
27. Covalently conjugated NOD2/TLR7 agonists are potent and versatile immune potentiatorsSamo Guzelj, Matjaž Weiss, Bram Slütter, Ruža Frkanec, Žiga Jakopin, 2022, izvirni znanstveni članek Ključne besede: immunostimulatory activity, vaccines, immune responses, pattern recognition receptors, synthesis of NOD2 agonist, Toll-like receptor 7 Celotno besedilo (datoteka, 4,87 MB) Gradivo ima več datotek! Več... |
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