1. Anthranilic acid inhibitors of undecaprenyl pyrophosphate synthase (UppS), an essential enzyme for bacterial cell wall biosynthesisMarko Jukič, Kaja Rožman, Matej Sova, Hélène Barreteau, Stanislav Gobec, 2019, izvirni znanstveni članek Ključne besede: UppS, inhibitors, cell-wall, pharmacophore model, antibacterial agents, undecaprenyl pyrophosphate synthase Celotno besedilo (datoteka, 4,42 MB) Gradivo ima več datotek! Več... |
2. Synthesis and evaluation of N-phenylpyrrolamides as DNA gyrase B inhibitorsMartina Durcik, Päivi Tammela, Michaela Barančokova, Tihomir Tomašič, Janez Ilaš, Danijel Kikelj, Nace Zidar, 2018, izvirni znanstveni članek Ključne besede: DNA gyrase, GyrB, antibacterials, inhibitors, pyrrolamides Celotno besedilo (datoteka, 452,68 KB) Gradivo ima več datotek! Več... |
3. Antimicrobial potencial of acinobacterial inhibotors of MurA and MurB ligases in bacterium Clostridium difficileElmedine Rustemi, 2019, magistrsko delo Ključne besede: molecular biology, cloning, Clostridium difficile, Mur ligases, actinobacterial inhibitors, protein expression, insect cells, purification, inhibitory assay Celotno besedilo (datoteka, 3,69 MB) |
4. Antimicrobial and modulatory activity of selected phytochemicals and epidemiological characteristics of antibiotic resistance in Camylobacter jejuniJasna Kovač, 2015, doktorska disertacija Ključne besede: Campylobacter jejuni, foodborne pathogens, antibiotic resistance, resistance modulation, plant extracts, pinocembrin, Alpinia katsumadai, essential oils, phytochemicals, alpha pinene, efflux inhibitors, adaptation response, epidemiology, MLST, gyr A typing, whole genome sequences, clonal expansion, campylobacteriosis prevalence, mathematical modelling Celotno besedilo (datoteka, 28,15 MB) |
5. DPP-4 inhibitors in the prevention/treatment of pulmonary fibrosis, heart and kidney injury caused by covid-19-a therapeutic approach of choice in type 2 diabetic patients?Andrija Smelcerović, Gordana Kocic, Mihajlo Gajic, Katarina Tomović, Vukica Djordjevic, Dobrila Stankovic-Djordjevic, Marko Anderluh, 2020, izvirni znanstveni članek Ključne besede: COVID-19, diabetes, DPP-4 inhibitors, fibrosis, multi-organ injury Celotno besedilo (datoteka, 375,34 KB) Gradivo ima več datotek! Več... |
6. Synthesis, molecular modelling and biological evaluation of novel heterodimeric, multiple ligands targeting cholinesterases and amyloid betaMichalina Hebda, Marek Bajda, Anna Więckowska, Natalia Szałaj, Anna Pasieka, Dawid Panek, Justyna Godyń, Tomasz Wichur, Damijan Knez, Stanislav Gobec, Barbara Malawska, 2016, izvirni znanstveni članek Ključne besede: cholinesterase inhibitors, molecular modelling, β-amyloid aggregation inhibitors, Alzheimer’s disease, multi-target-directed ligands (MTDL), PAMPA-BBB assay Celotno besedilo (datoteka, 3,87 MB) Gradivo ima več datotek! Več... |
7. Synthesis and biological evaluation of benzochromenopyrimidinones as cholinesterase inhibitors and potent antioxidant, non-hepatotoxic agents for Alzheimer's diseaseYoussef Dgachi, Oscar M. Bautista-Aguilera, Mohamed Benchekroun, Hélène Martin, Alexandre Bonet, Damijan Knez, Justyna Godyń, Barbara Malawska, Stanislav Gobec, Mourad Chioua, Jana Janockova, Ondrej Soukup, Fakher Chabchoub, José Marco-Contelles, Lhassane Ismaili, 2016, izvirni znanstveni članek Ključne besede: Alzheimer's disease, quinazolinones, multicomponent reactions, multitarget-directed ligands, antioxidants, cholinesterase inhibitors, hepatotoxicity Celotno besedilo (datoteka, 1,47 MB) Gradivo ima več datotek! Več... |
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9. Design, synthesis, and biological evaluation of 2-(benzylamino-2-hydroxyalkyl)isoindoline-1,3-diones derivatives as potential disease-modifying multifunctional anti-Alzheimer agentsDawid Panek, Anna Więckowska, Anna Pasieka, Justyna Godyń, Jakub Jończyk, Marek Bajda, Damijan Knez, Stanislav Gobec, Barbara Malawska, 2018, izvirni znanstveni članek Ključne besede: isoindoline-1, 3-dione derivatives, cholinesterase inhibitors, BACE-1 inhibitors, Aβ-aggregation, molecular modeling, multiple anti-Alzheimer's ligands Celotno besedilo (datoteka, 6,29 MB) Gradivo ima več datotek! Več... |
10. Early Lyme borreliosis in patients treated with tumour necrosis factor-alfa inhibitorsVera Maraspin-Čarman, Petra Bogovič, Tereza Rojko, Katarina Ogrinc, Eva Ružić-Sabljić, Franc Strle, 2019, izvirni znanstveni članek Ključne besede: Lyme borreliosis, immunocompromised host, TNF-α inhibitors, erythema migrans, treatment, outcome Celotno besedilo (datoteka, 234,57 KB) Gradivo ima več datotek! Več... |