31. Echinacea angustifolia DC. lipophilic extract patch for skin applicationDritan Hasa, Simon Žakelj, Iztok Grabnar, Francesco Cilurzo, Stefano Dall'Acqua, Antonella Riva, Beatrice Perissutti, Dario Voinovich, 2020, izvirni znanstveni članek Ključne besede: Echinacea angustifolia lipophilic extract, tetraene, drug-in-adhesive patch, in vitro skin permeation, pharmacokinetics Celotno besedilo (datoteka, 1,40 MB) Gradivo ima več datotek! Več... |
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34. Analytical techniques for structural characterization of proteins in solid pharmaceutical formsAljoša Bolje, Stanislav Gobec, 2021, pregledni znanstveni članek Ključne besede: solid pharmaceuticals, lyophilization, analytical tools, protein characterization, protein structure, formulation development, antibody, excipients, stable drug product, safe drug Celotno besedilo (datoteka, 7,49 MB) Gradivo ima več datotek! Več... |
35. Prioritisation of compounds for 3CL$^{pro}$ inhibitor development on SARS-CoV-2 variantsMarko Jukič, Blaž Škrlj, Gašper Tomšič, Sebastian Pleško, Črtomir Podlipnik, Urban Bren, 2021, izvirni znanstveni članek Ključne besede: COVID-19, SARS-CoV-2, free-energy calculations, in silico drug design, virtual screening, inhibitors, 3C-like protease, M$^{pro}$, 3CL$^{pro}$, high-throughput, chemical library design, machine learning, compound prioritisation Celotno besedilo (datoteka, 6,56 MB) Gradivo ima več datotek! Več... |
36. Computational design and development of benzodioxane-benzamides as potent inhibitors of FtsZ by exploring the hydrophobic subpocketValentina Straniero, Victor Sebastián-Pérez, Lorenzo Suigo, William Margolin, Andrea Casiraghi, Martina Hrast, Carlo Zanotto, Irena Zdovc, Antonia Radaelli, Ermanno Valoti, 2021, izvirni znanstveni članek Ključne besede: gram positive-dependent diseases, antibiotic-resistance, MSSA, MRSA, Bacillus subtilis, FtsZ, Z ring, FtsZ inhibition, MIC, pharmacology, chemistry, anti-bacterial agents, methicillin-resistant Staphylococcus aureus, drug resistance, microbiology, benzamides, bacterial proteins Celotno besedilo (datoteka, 5,49 MB) Gradivo ima več datotek! Več... |
37. Nanotechnology-based drug delivery to improve the therapeutic benefits of NRF2 modulators in cancer therapyZerrin Sezgin-Bayindir, Sonia Losada-Barreiro, Carlos Bravo-Díaz, Matej Sova, Julijana Kristl, Luciano Saso, 2021, pregledni znanstveni članek Ključne besede: NRF2 modulators, anticancer agents, nanoparticles, drug delivery, drug targeting Celotno besedilo (datoteka, 1,96 MB) Gradivo ima več datotek! Več... |
38. Targeted cancer therapy using compounds activated by lightPetra Dunkel, Janez Ilaš, 2021, pregledni znanstveni članek Ključne besede: photocages, photoswitches, photopharmacology, light-activatable materials, photoresponsive drug delivery systems, azobenzenes Celotno besedilo (datoteka, 8,51 MB) Gradivo ima več datotek! Več... |
39. Metronomic chemotherapy for palliative treatment of malignant oral tumors in dogsNina Milevoj, Ana Nemec, Nataša Tozon, 2022, izvirni znanstveni članek Ključne besede: metronomic chemotherapy, cyclophosphamide, malignant oral tumors, dogs, palliative treatment, drug therapy, neoplasms, palliative care Celotno besedilo (datoteka, 563,76 KB) Gradivo ima več datotek! Več... |
40. A fine-tuned lipophilicity/hydrophilicity ratio governs antibacterial potency and selectivity of bifurcated halogen bond-forming NBTIsAnja Kolarič, Maja Kokot, Martina Hrast, Matjaž Weiss, Irena Zdovc, Jurij Trontelj, Simon Žakelj, Marko Anderluh, Nikola Minovski, 2021, izvirni znanstveni članek Ključne besede: antibacterials, drug discovery, DNA gyrase inhibitors, topoisomerase IV inhibitors, intercalators, novel bacterial topoisomerase inhibitors, topoisomerase II inhibitors, intercalating agents Celotno besedilo (datoteka, 6,80 MB) Gradivo ima več datotek! Več... |