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182. Synthesis, molecular modelling and biological evaluation of novel heterodimeric, multiple ligands targeting cholinesterases and amyloid betaMichalina Hebda, Marek Bajda, Anna Więckowska, Natalia Szałaj, Anna Pasieka, Dawid Panek, Justyna Godyń, Tomasz Wichur, Damijan Knez, Stanislav Gobec, Barbara Malawska, 2016, izvirni znanstveni članek Ključne besede: cholinesterase inhibitors, molecular modelling, β-amyloid aggregation inhibitors, Alzheimer’s disease, multi-target-directed ligands (MTDL), PAMPA-BBB assay Celotno besedilo (datoteka, 3,87 MB) Gradivo ima več datotek! Več... |
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184. Discovery of immunoproteasome inhibitors using large-scale covalent virtual screeningAndrea Scarpino, Dávid Bajusz, Matic Proj, Martina Gobec, Izidor Sosič, Stanislav Gobec, György G. Ferenczy, György Keserü M., 2019, izvirni znanstveni članek Ključne besede: immunoproteasome, covalent inhibitor, virtual screening, β5i selective inhibitor Celotno besedilo (datoteka, 3,77 MB) Gradivo ima več datotek! Več... |
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186. Bromo-cyclobutenaminones as new covalent UDP-N-acetylglucosamine enolpyruvyl transferase (MurA) inhibitorsDavid J. Hamilton, Péter Ábrányi-Balogh, Aaron Keeley, László Petri, Martina Hrast, Tímea Imre, Maikel Wijtmans, Stanislav Gobec, Iwan J. P. de Esch, György Keserü M., 2020, izvirni znanstveni članek Ključne besede: covalent inhibitor, MurA, cyclobutenaminone, antibacterial, irreversible Celotno besedilo (datoteka, 1,08 MB) Gradivo ima več datotek! Več... |
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