1. Benzamide derivatives targeting the cell division protein FtsZValentina Straniero, Lorenzo Suigo, Andrea Casiraghi, Victor Sebastián-Pérez, Martina Hrast, Carlo Zanotto, Irena Zdovc, Carlo De Giuli Morghen, Antonia Radaelli, Ermanno Valoti, 2020, izvirni znanstveni članek Ključne besede: cell division protein FtsZ, benzamide, 1, 4-benzodioxane, 1, 4-benzoxathiane, multi-drug resistant Staphylococcus aureus, Escherichia coli N43, veterinary medicine Celotno besedilo (datoteka, 6,25 MB) Gradivo ima več datotek! Več... |
2. Synthesis and evaluation of antioxidant properties of 2-substituted quinazolin-4(3H)-onesJanez Mravljak, Lara Slavec, Martina Hrast, Matej Sova, 2021, izvirni znanstveni članek Ključne besede: quinazolinone, synthesis, antioxidant, DPPH, ABTS, CUPRAC, metal-chelating properties Celotno besedilo (datoteka, 2,84 MB) Gradivo ima več datotek! Več... |
3. Amide containing NBTI antibacterials with reduced hERG inhibition, retained antimicrobial activity against gram-positive bacteria and in vivo efficacyMaja Kokot, Matjaž Weiss, Irena Zdovc, Lidija Senerovic, Natasa Radakovic, Marko Anderluh, Nikola Minovski, Martina Hrast, 2023, izvirni znanstveni članek Ključne besede: NBTIs, DNA gyrase, topoisomerase IV, antibacterials, MRSA, hERG inhibition, in vivo efficacy Celotno besedilo (datoteka, 3,61 MB) Gradivo ima več datotek! Več... |
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5. Inhibition of MurA enzyme from Escherichia coli and Staphylococcus aureus by diterpenes from Lepechinia meyenii and their synthetic analogsMacarena Funes Chabán, Martina Hrast, Rok Frlan, Dafni G. Graikioti, Constantinos M. Athanassopoulos, María Cecilia Carpinella, 2021, izvirni znanstveni članek Ključne besede: dehydroabietane derivatives, diterpenes, MurA inhibitors, MurF inhibitors, Staphylococcus aureus MurA, Escherichia coli MurA Celotno besedilo (datoteka, 2,12 MB) Gradivo ima več datotek! Več... |
6. Potent DNA gyrase inhibitors bind asymmetrically to their target using symmetrical bifurcated halogen bondsAnja Kolarič, Thomas Germe, Martina Hrast, Clare E. M. Stevenson, David M. Lawson, Nicolas P. Burton, Judit Vörös, Anthony Maxwell, Nikola Minovski, Marko Anderluh, 2021, izvirni znanstveni članek Ključne besede: antibacterials, DNA gyrase inhibitors, drug discovery, Staphylococcus aureus, intercalators, novel bacterial topoisomerase inhibitors, NBTIs, symmetrical bifurcated halogen bonds, crystal structure, novel NBTIs mechanism of action, antimicrobials, DNA-binding proteins, drug development, X-ray crystallography Celotno besedilo (datoteka, 2,00 MB) Gradivo ima več datotek! Več... |
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9. DNA-encoded library screening on two validated enzymes of the peptidoglycan biosynthetic pathwayMatic Proj, Krištof Bozovičar, Martina Hrast, Rok Frlan, Stanislav Gobec, 2022, izvirni znanstveni članek Ključne besede: antibacterial agents, DNA-encoded library, screening, inhibitors Celotno besedilo (datoteka, 1,04 MB) Gradivo ima več datotek! Več... |
10. Bromo-cyclobutenaminones as new covalent UDP-N-acetylglucosamine enolpyruvyl transferase (MurA) inhibitorsDavid J. Hamilton, Péter Ábrányi-Balogh, Aaron Keeley, László Petri, Martina Hrast, Tímea Imre, Maikel Wijtmans, Stanislav Gobec, Iwan J. P. de Esch, György Keserü M., 2020, izvirni znanstveni članek Ključne besede: covalent inhibitor, MurA, cyclobutenaminone, antibacterial, irreversible Celotno besedilo (datoteka, 1,08 MB) Gradivo ima več datotek! Več... |