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1. Next-generation heterocyclic electrophiles as small-molecule covalent MurA inhibitors Péter Ábrányi-Balogh, Aaron Keeley, György G. Ferenczy, László Petri, Tímea Imre, Katarina Grabrijan, Martina Hrast, Damijan Knez, Janez Ilaš, Stanislav Gobec, György Keserü M., 2022, izvirni znanstveni članek Ključne besede: covalent inhibitor, heterocyclic electrophiles, cysteine labelling, quaternization, MurA |
2. Bromo-cyclobutenaminones as new covalent UDP-N-acetylglucosamine enolpyruvyl transferase (MurA) inhibitors David J. Hamilton, Péter Ábrányi-Balogh, Aaron Keeley, László Petri, Martina Hrast, Tímea Imre, Maikel Wijtmans, Stanislav Gobec, Iwan J. P. de Esch, György Keserü M., 2020, izvirni znanstveni članek Ključne besede: covalent inhibitor, MurA, cyclobutenaminone, antibacterial, irreversible |