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1. Structure-activity relationships of benzothiazole-based Hsp90 C-terminal-domain inhibitors Jaka Dernovšek, Živa Zajec, Martina Durcik, Lucija Peterlin-Mašič, Martina Gobec, Nace Zidar, Tihomir Tomašič, 2021, original scientific article Keywords: allostery, Hsp90, benzothiazole, cancer, inhibitor, cancer therapy |
2. Exploring the chemical space of benzothiazole-based DNA gyrase B inhibitors Žiga Skok, Michaela Barančokova, Ondřej Benek, Cristina Durante Cruz, Päivi Tammela, Tihomir Tomašič, Nace Zidar, Lucija Peterlin-Mašič, Anamarija Zega, Danijel Kikelj, Janez Ilaš, 2020, original scientific article Keywords: DNA gyrase, topoisomerase IV, GyrB, ParE, antibacterial benzothiazole |