31. Inhibition of the SARS-CoV-2 3CL$^{pro}$ main protease by plant polyphenolsMiha Bahun, Marko Jukič, Domen Oblak, Luka Kranjc, Gregor Bajc, Matej Butala, Krištof Bozovičar, Tomaž Bratkovič, Črtomir Podlipnik, Nataša Poklar Ulrih, 2022, original scientific article Keywords: edible plants, polyphenols, COVID-19, SARS-CoV-2, 3CL$^{pro}$, protease inhibitor Full text (file, 2,14 MB) This document has more files! More... |
32. Structural isomerism and enhanced lipophilicity of pyrithione ligands of organoruthenium(II) complexes increase inhibition on AChE and BuChEJerneja Kladnik, Samuel Ristovski, Jakob Kljun, Andrea Defant, Ines Mancini, Kristina Sepčić, Iztok Turel, 2020, original scientific article Keywords: Alzheimer’s disease, acetylcholinesterase, butyrylcholinesterase, cholinesterase inhibitor, molecular docking, organoruthenium(II) complexes, pyrithione derivatives Full text (file, 1,28 MB) This document has more files! More... |
33. Discovery of novel Hsp90 C-terminal inhibitors using 3D-pharmacophores derived from molecular dynamics simulationsTihomir Tomašič, Martina Durcik, Bradley M. Keegan, Darja Gramec, Živa Zajec, Brian S. J. Blagg, Sharon D. Bryant, 2020, original scientific article Keywords: allosteric, cancer, Hsp90, inhibitor, molecular dynamics, pharmacophores, virtual screening Full text (file, 7,84 MB) This document has more files! More... |
34. Bromo-cyclobutenaminones as new covalent UDP-N-acetylglucosamine enolpyruvyl transferase (MurA) inhibitorsDavid J. Hamilton, Péter Ábrányi-Balogh, Aaron Keeley, László Petri, Martina Hrast, Tímea Imre, Maikel Wijtmans, Stanislav Gobec, Iwan J. P. de Esch, György Keserü M., 2020, original scientific article Keywords: covalent inhibitor, MurA, cyclobutenaminone, antibacterial, irreversible Full text (file, 1,08 MB) This document has more files! More... |
35. Hybrid inhibitors of DNA gyrase A and BMartina Durcik, Žiga Skok, Janez Ilaš, Nace Zidar, Anamarija Zega, Petra Szili, Gábor Draskovits, T. Revesz, Danijel Kikelj, Ákos Nyerges, Csaba Pál, Lucija Peterlin-Mašič, Tihomir Tomašič, 2021, original scientific article Keywords: antibacterial, ciprofloxacin, DNA gyrase, dual inhibitor, hybrid Full text (file, 3,42 MB) This document has more files! More... |
36. Overview of the assays to probe O-linked β-N-acetylglucosamine transferase binding and activityCyril Balsollier, Roland J. Pieters, Marko Anderluh, 2021, review article Keywords: OGT, GlcNAcylation, O-GlcNAc transferase, bioassay, OGT inhibitor Full text (file, 5,14 MB) This document has more files! More... |
37. Structure-activity relationships of benzothiazole-based Hsp90 C-terminal-domain inhibitorsJaka Dernovšek, Živa Zajec, Martina Durcik, Lucija Peterlin-Mašič, Martina Gobec, Nace Zidar, Tihomir Tomašič, 2021, original scientific article Keywords: allostery, Hsp90, benzothiazole, cancer, inhibitor, cancer therapy Full text (file, 7,92 MB) This document has more files! More... |
38. Efflux pump inhibition and resistance modulation in Mycobacterium smegmatis by Peucedanum ostruthium and its coumarinsKatarina Šimunović, Julia Solnier, Fabian Alperth, Olaf Kunert, Sonja Smole Možina, Franz Bucar, 2021, original scientific article Keywords: Mycobacterium smegmatis, efflux pump inhibitor, Peucedanum ostruthium, antibacterial properties, ostruthin, imperatorin, ethidium bromide accumulation, resistance modulation Full text (file, 2,08 MB) This document has more files! More... |
39. Overview of immune checkpoint inhibitors in gynecological cancer treatmentBoštjan Pirš, Erik Škof, Vladimir Smrkolj, Špela Smrkolj, 2022, review article Keywords: immune check-point inhibitor, biomarker, endometrial cancer, ovarian cancer, uterine cervical cancer, vulvar cancer, treatment response prediction Full text (file, 731,71 KB) This document has more files! More... |
40. Association of myocardial infarction with CDKN2B Antisense RNA 1 (CDKN2B-AS1) rs1333049 polymorphism in Slovenian subjects with type 2 diabetes mellitusMiha Tibaut, Franjo Naji, Danijel Petrovič, 2022, original scientific article Keywords: type 2 diabetes mellitus, myocardial infarction, coronary artery disease, Cyclin Dependent Kinase Inhibitor 2B Antisense RNA 1, CDKN2B-AS1, rs1333049 Full text (file, 229,89 KB) This document has more files! More... |