1. Anthranilic acid inhibitors of undecaprenyl pyrophosphate synthase (UppS), an essential enzyme for bacterial cell wall biosynthesisMarko Jukič, Kaja Rožman, Matej Sova, Hélène Barreteau, Stanislav Gobec, 2019, original scientific article Keywords: UppS, inhibitors, cell-wall, pharmacophore model, antibacterial agents, undecaprenyl pyrophosphate synthase
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2. DNA-encoded library screening on two validated enzymes of the peptidoglycan biosynthetic pathwayMatic Proj, Krištof Bozovičar, Martina Hrast, Rok Frlan, Stanislav Gobec, 2022, original scientific article Keywords: antibacterial agents, DNA-encoded library, screening, inhibitors
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3. Covalent inhibitors of bacterial peptidoglycan biosynthesis enzyme MurA with chloroacetamide warheadKatarina Grabrijan, Martina Hrast, Matic Proj, Ana Dolšak, Irena Zdovc, Tímea Imre, László Petri, Péter Ábrányi-Balogh, György Keserü M., Stanislav Gobec, 2022, original scientific article Keywords: antibacterial agents, UDP-N-acetylglucosamine enolpyruvyl transferase, thiol reactivity
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4. The synthesis of (2R)-aziridine-2-carboxylic acid containing dipeptidesSamo Kuzmič, Martina Hrast, Rok Frlan, 2022, original scientific article Keywords: dipeptides, aziridines, biomarkers, warheads, antibacterial agents
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5. Discovery of a fragment hit compound targeting D-Ala:D-Ala ligase of bacterial peptidoglycan biosynthesisMatic Proj, Martina Hrast, Gregor Bajc, Rok Frlan, Anže Meden, Matej Butala, Stanislav Gobec, 2023, original scientific article Keywords: fragment-based drug discovery, hit triage, inhibitors, antibacterial agents
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6. Improved N-phenylpyrrolamide inhibitors of DNA gyrase as antibacterial agents for high-priority bacterial strainsNace Zidar, Alessia Onali, Peter Peršolja, Davide Benedetto Tiz, Jaka Dernovšek, Žiga Skok, Martina Durcik, Andrej Emanuel Cotman, Martina Hrast, Anamarija Zega, Lucija Peterlin-Mašič, Janez Ilaš, Tihomir Tomašič, Danijel Kikelj, 2024, original scientific article Keywords: antibacterial agents, DNA gyrase, GyrB, inhibitor, N-phenylpyrrolamide, ParE, topoisomerase IV
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7. Synthesis and biochemical evaluation of new 3-amido-4-substituted monocyclic ß-lactams as inhibitors of penicillin-binding protein(s)Katarina Grabrijan, Nika Strašek Benedik, Alen Krajnc, Krištof Bozovičar, Damijan Knez, Matic Proj, Irena Zdovc, Izidor Sosič, Martina Hrast, Stanislav Gobec, 2024, original scientific article Keywords: antibacterial agents, monocyclic-β-lactams, penicillin-binding proteins, covalent inhibitors, transpeptidase
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