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8. Discovery of a new drug-like series of OGT inhibitors by virtual screeningElena Maria Loi, Tihomir Tomašič, Cyril Balsollier, Kevin van Eekelen, Matjaž Weiss, Martina Gobec, Matthew G Alteen, David J. Vocadlo, Roland J. Pieters, Marko Anderluh, 2022, original scientific article Keywords: O-GlcNAc transferase, OGT inhibitors, virtual screening, pharmaceutical chemistry Full text (file, 10,66 MB) This document has more files! More... |
9. Strukturno podprto načrtovanje, sinteza in biološko vrednotenje novih zaviralcev O-β-N-acetilglukozaminil transferazeElena Maria Loi, 2023, doctoral dissertation Keywords: O-GlcNAcylation, OGT, OGA, OGT inhibitors, posttranslational, modifications, computational drug design, virtual screening, ester hydrolysis, metabolic stability Full text (file, 20,68 MB) |
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