1. Antimicrobial activity of the marine alkaloids, clathrodin and oroidin, and their synthetic analoguesNace Zidar, Sofia Montalvão, Žiga Hodnik, Dorota A. Nawrot, Aleš Žula, Janez Ilaš, Danijel Kikelj, Päivi Tammela, Lucija Peterlin-Mašič, 2014, original scientific article Keywords: marine alkaloid, Agelas, antimicrobial, antibacterial, antifungal, pyrrole-2-aminoimidazole, oroidin, clathrodin
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3. Synthesis and evaluation of N-phenylpyrrolamides as DNA gyrase B inhibitorsMartina Durcik, Päivi Tammela, Michaela Barančokova, Tihomir Tomašič, Janez Ilaš, Danijel Kikelj, Nace Zidar, 2018, original scientific article Keywords: DNA gyrase, GyrB, antibacterials, inhibitors, pyrrolamides
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4. Design, synthesis and biological evaluation of 4,5-dibromo-N-(thiazol-2-yl)-1H-pyrrole-2-carboxamide derivatives as novel DNA gyrase inhibitorsTihomir Tomašič, Matic Mirt, Michaela Barančokova, Janez Ilaš, Nace Zidar, Päivi Tammela, Danijel Kikelj, 2017, original scientific article Keywords: antibacterial, DNA gyrase, docking, inhibitor, thiazole
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5. Discovery of substituted oxadiazoles as a novel scaffold for DNA gyrase inhibitorsŽiga Jakopin, Janez Ilaš, Michaela Barančokova, Matjaž Brvar, Päivi Tammela, Marija Sollner Dolenc, Tihomir Tomašič, Danijel Kikelj, 2017, original scientific article Keywords: 1, 2, 4-oxadiazoles, DNA gyrase inhibition, topoisomerase IV inhibition, antibacterial screening, computer-aided drug design
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6. Discovery of benzothiazole scaffold-based DNA gyrase B inhibitorsMarina Gjorgjieva, Tihomir Tomašič, Michaela Barančokova, Sotirios Katsamakas, Janez Ilaš, Päivi Tammela, Lucija Peterlin-Mašič, Danijel Kikelj, 2016, original scientific article Keywords: organoruthenium complexes, diketonates, anticancer drugs, ROS, cytotoxicity, cell cycle arrest
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7. Exploring the chemical space of benzothiazole-based DNA gyrase B inhibitorsŽiga Skok, Michaela Barančokova, Ondřej Benek, Cristina Durante Cruz, Päivi Tammela, Tihomir Tomašič, Nace Zidar, Lucija Peterlin-Mašič, Anamarija Zega, Danijel Kikelj, Janez Ilaš, 2020, original scientific article Keywords: DNA gyrase, topoisomerase IV, GyrB, ParE, antibacterial benzothiazole
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