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22. Structure-activity relationships of benzothiazole-based Hsp90 C-terminal-domain inhibitorsJaka Dernovšek, Živa Zajec, Martina Durcik, Lucija Peterlin-Mašič, Martina Gobec, Nace Zidar, Tihomir Tomašič, 2021, original scientific article Keywords: allostery, Hsp90, benzothiazole, cancer, inhibitor, cancer therapy Full text (file, 7,92 MB) This document has more files! More... |
23. Neuroinflammation-induced upregulation of glial cathepsin X expression and activity in vivoAnja Pišlar, Larisa Tratnjek, Gordana Glavan, Nace Zidar, Marko Živin, Janko Kos, 2020, original scientific article Keywords: neuroinflammation, neurodegeneration, lipopolysaccharide, glia, cathepsin X, neuroprotection Full text (file, 7,62 MB) This document has more files! More... |
24. ATP-competitive inhibitors of human DNA topoisomerase IIα with improved antiproliferative activity based on N-phenylpyrrolamide scaffoldŽiga Skok, Martina Durcik, Živa Zajec, Darja Gramec, Krištof Bozovičar, Anja Pišlar, Tihomir Tomašič, Anamarija Zega, Lucija Peterlin-Mašič, Danijel Kikelj, Nace Zidar, Janez Ilaš, 2023, original scientific article Keywords: anticancer drugs, ATP-competitive inhibitors, catalytic inhibitor, cytotoxicity, human DNA topoisomerase II Full text (file, 2,83 MB) This document has more files! More... |
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27. Sinteza in vrednotenje novih N-(4-karbamoilfenil)pirolamidnih zaviralcev človeške DNA-topoizomeraze IINataša Turk, 2019, master's thesis Keywords: DNA-topoizomeraza II, protirakave učinkovine, ATP-kompetitivni zaviralci, N-(4-karbamoilfenil)pirolamidi, zaviralci angiogeneze, zaviralci sinteze DNA, sinteza spojin, sintezni postopki Full text (file, 1,59 MB) |
28. Sinteza 5-fenil-1,5-dihidro-pirano [2,3-d]pirimidin-2,4-dionov in 5-benzoilpirimidin-2,4,6-trionov ter vrednotenje njihovih antioksidativnih lastnostiAna Čelhar, 2017, undergraduate thesis Keywords: prosti radikali, antioksidanti, 1, 1-difenil-2-pikrilhidrazil, 5-benzoilpirimidin-2, 4, 6-trion, barbiturna kislina, 5-fenil-1, 5-dihidro-pirano [2, 3-d]pirimidin-2.4-dion Full text (outside link) |
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30. Antimicrobial activity of the marine alkaloids, clathrodin and oroidin, and their synthetic analoguesNace Zidar, Sofia Montalvão, Žiga Hodnik, Dorota A. Nawrot, Aleš Žula, Janez Ilaš, Danijel Kikelj, Päivi Tammela, Lucija Peterlin-Mašič, 2014, original scientific article Keywords: marine alkaloid, Agelas, antimicrobial, antibacterial, antifungal, pyrrole-2-aminoimidazole, oroidin, clathrodin Full text (file, 935,08 KB) This document has more files! More... |