1. Recent progress in the discovery and development of DNA gyrase B inhibitorsMichaela Barančokova, Danijel Kikelj, Janez Ilaš, 2018, review article Keywords: antibacterial, ATP-competitive, DNA gyrase, drug discovery, Gram-negative bacteria, GyrB, inhibitor, Par, topoisomerase II, topoisomerase IV Full text (file, 717,37 KB) This document has more files! More... |
2. Discovery of substituted oxadiazoles as a novel scaffold for DNA gyrase inhibitorsŽiga Jakopin, Janez Ilaš, Michaela Barančokova, Matjaž Brvar, Päivi Tammela, Marija Sollner Dolenc, Tihomir Tomašič, Danijel Kikelj, 2017, original scientific article Keywords: 1, 2, 4-oxadiazoles, DNA gyrase inhibition, topoisomerase IV inhibition, antibacterial screening, computer-aided drug design Full text (file, 1,45 MB) This document has more files! More... |
3. Design, synthesis and biological evaluation of 4,5-dibromo-N-(thiazol-2-yl)-1H-pyrrole-2-carboxamide derivatives as novel DNA gyrase inhibitorsTihomir Tomašič, Matic Mirt, Michaela Barančokova, Janez Ilaš, Nace Zidar, Päivi Tammela, Danijel Kikelj, 2017, original scientific article Keywords: antibacterial, DNA gyrase, docking, inhibitor, thiazole Full text (file, 1,60 MB) This document has more files! More... |
4. Synthesis and evaluation of N-phenylpyrrolamides as DNA gyrase B inhibitorsMartina Durcik, Päivi Tammela, Michaela Barančokova, Tihomir Tomašič, Janez Ilaš, Danijel Kikelj, Nace Zidar, 2018, original scientific article Keywords: DNA gyrase, GyrB, antibacterials, inhibitors, pyrrolamides Full text (file, 452,68 KB) This document has more files! More... |
5. Discovery of benzothiazole scaffold-based DNA gyrase B inhibitorsMarina Gjorgjieva, Tihomir Tomašič, Michaela Barančokova, Sotirios Katsamakas, Janez Ilaš, Päivi Tammela, Lucija Peterlin-Mašič, Danijel Kikelj, 2016, original scientific article Keywords: organoruthenium complexes, diketonates, anticancer drugs, ROS, cytotoxicity, cell cycle arrest Full text (file, 1,17 MB) This document has more files! More... |
6. Exploring the chemical space of benzothiazole-based DNA gyrase B inhibitorsŽiga Skok, Michaela Barančokova, Ondřej Benek, Cristina Durante Cruz, Päivi Tammela, Tihomir Tomašič, Nace Zidar, Lucija Peterlin-Mašič, Anamarija Zega, Danijel Kikelj, Janez Ilaš, 2020, original scientific article Keywords: DNA gyrase, topoisomerase IV, GyrB, ParE, antibacterial benzothiazole Full text (file, 2,22 MB) This document has more files! More... |
7. Exploring the interaction of N-(benzothiazol-2-yl)pyrrolamide DNA gyrase inhibitors with the GyrB ATP-binding site lipophilic floorNace Zidar, Andrej Emanuel Cotman, Wessel Sinnige, Ondřej Benek, Michaela Barančokova, Anamarija Zega, Lucija Peterlin-Mašič, Tihomir Tomašič, Janez Ilaš, Ricardo D. Enriz, Danijel Kikelj, 2024, original scientific article Keywords: antibacterial agent, DNA gyrase, ATP-binding site, N-(benzothiazol-2-yl)pyrrolamide, inhibitor, QTAIM analysis Full text (file, 2,64 MB) This document has more files! More... |