1. Sinteza 4,5,6,7-tetrahidrobenzotiazolnih zaviralcev C-končne domene proteina toplotnega šoka 90Maja Mavri, 2022, master's thesis/paper Keywords: Hsp90, rak, zaviralci C-končne domene, 4, 5, 6, 7-tetrahidrobenzotiazol, 3, 4-diklorofenil, SAR Full text (file, 1,91 MB) |
2. Načrtovanje, sinteza in vrednotenje 1,4-disubstituiranih-1,2,3-triazolo-galaktozidov kot zaviralcev galektinov-1 in -8Jaka Dernovšek, 2020, master's thesis/paper Keywords: galaktoza, galektin-1, galektin-8, SAR, selektivnost, sidranje Full text (file, 2,35 MB) |
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4. Sinteza 4,5,6,7-tetrahidrobenzotiazolnih alosteričnih zaviralcev proteina toplotnega šoka 90Svit Ferjančič Benetik, 2021, master's thesis/paper Keywords: Hsp90, 4, 5, 6, 7-tetrahidrobenzotiazol, C-končna domena, SAR, rak Full text (file, 2,14 MB) |
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8. Structure-activity relationships of benzothiazole-based Hsp90 C-terminal-domain inhibitorsJaka Dernovšek, Živa Zajec, Martina Durcik, Lucija Peterlin-Mašič, Martina Gobec, Nace Zidar, Tihomir Tomašič, 2021, original scientific article Keywords: allostery, Hsp90, benzothiazole, cancer, inhibitor, cancer therapy Full text (file, 7,92 MB) This document has more files! More... |
9. Design and synthesis of novel 3-triazolyl-1-thiogalactosides as galectin-1, -3 and -8 inhibitorsSjors van Klaveren, Jaka Dernovšek, Žiga Jakopin, Marko Anderluh, Hakon Leffler, Ulf Nilsson, Tihomir Tomašič, 2022, original scientific article Full text (file, 1010,75 KB) This document has more files! More... |
10. In silico discovery and optimisation of a novel structural class of Hsp90 C-terminal domain inhibitorsŽiva Zajec, Jaka Dernovšek, Martina Gobec, Tihomir Tomašič, 2022, original scientific article Keywords: allosteric, cancer, heat shock, Hsp90, inhibitor, virtual screening Full text (file, 7,89 MB) This document has more files! More... |