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6. Načrtovanje, sinteza in biološko vrednotenje novih alosteričnih zaviralcev Hsp90 s protitumornim delovanjemŽiva Zajec, 2023, doctoral dissertation Keywords: Hsp90, rak, zaviralci, alosterični, virtualno rešetanje, molekulsko modeliranje Full text (file, 35,52 MB) |
7. Discovery of novel Hsp90 C-terminal inhibitors using 3D-pharmacophores derived from molecular dynamics simulationsTihomir Tomašič, Martina Durcik, Bradley M. Keegan, Darja Gramec, Živa Zajec, Brian S. J. Blagg, Sharon D. Bryant, 2020, original scientific article Keywords: allosteric, cancer, Hsp90, inhibitor, molecular dynamics, pharmacophores, virtual screening Full text (file, 7,84 MB) This document has more files! More... |
8. Structure-activity relationships of benzothiazole-based Hsp90 C-terminal-domain inhibitorsJaka Dernovšek, Živa Zajec, Martina Durcik, Lucija Peterlin-Mašič, Martina Gobec, Nace Zidar, Tihomir Tomašič, 2021, original scientific article Keywords: allostery, Hsp90, benzothiazole, cancer, inhibitor, cancer therapy Full text (file, 7,92 MB) This document has more files! More... |
9. Exploration and optimisation of structure-activity relationships of new triazole-based C-terminal Hsp90 inhibitors towards in vivo anticancer potencyJaka Dernovšek, Živa Zajec, Dunja Urbančič, Irena Mlinarič-Raščan, Andrej Emanuel Cotman, Nace Zidar, Tihomir Tomašič, 2024, original scientific article Keywords: cancer, Hsp90, inhibitor, Ewing sarcoma, zebrafish Full text (file, 8,03 MB) This document has more files! More... |
10. ATP-competitive inhibitors of human DNA topoisomerase IIα with improved antiproliferative activity based on N-phenylpyrrolamide scaffoldŽiga Skok, Martina Durcik, Živa Zajec, Darja Gramec, Krištof Bozovičar, Anja Pišlar, Tihomir Tomašič, Anamarija Zega, Lucija Peterlin-Mašič, Danijel Kikelj, Nace Zidar, Janez Ilaš, 2023, original scientific article Keywords: anticancer drugs, ATP-competitive inhibitors, catalytic inhibitor, cytotoxicity, human DNA topoisomerase II Full text (file, 2,83 MB) This document has more files! More... |