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1. Evaluation of firefly and Renilla luciferase inhibition in reporter-gene assays Maša Kenda, Jan Vegelj, Barbara Herlah, Andrej Perdih, Přemysl Mladěnka, Marija Sollner Dolenc, 2021, original scientific article Keywords: isoflavonoids, firefly luciferase, Renilla luciferase, inhibition, quantitative structure–activity relationships, molecular docking, reporter-gene assay, OECD test guidelines, alternative methods |
2. Synthesis and evaluation of AKR1C inhibitory properties of A-ring halogenated oestrone derivatives Maša Sinreih, Rebeka Jójárt, Zoltán Kele, Tomaž Büdefeld, Gábor Paragi, Erzsébet Mernyák, Tea Lanišnik-Rižner, 2021, original scientific article Keywords: aldo-keto reductases, inhibition, halogenated oestrone derivatives, structure–activity relationships |