1. 3D pharmacophore-based discovery of novel Kv10.1 inhibitors with antiproliferative activityŽan Toplak, Louise Antonia Hendrickx, Špela Gubič, Štefan Možina, Bojana Žegura, Alja Štern, Matjaž Novak, Xiaoyi Shi, Steve Peigneur, Jan Tytgat, Tihomir Tomašič, Luis A. Pardo, Lucija Peterlin-Mašič, 2021, original scientific article Keywords: K$_V$10.1, ion channels, hERG, pharmacophore modelling, virtual screening, antiproliferative activity Full text (file, 14,79 MB) This document has more files! More... |
2. New diarylamine KV10.1 inhibitors and their anticancer potentialŠpela Gubič, Žan Toplak, Xiaoyi Shi, Jaka Dernovšek, Louise Antonia Hendrickx, Ernesto Lopes Pinheiro-Junior, Steve Peigneur, Jan Tytgat, Luis A. Pardo, Lucija Peterlin-Mašič, Tihomir Tomašič, 2022, original scientific article Keywords: KV10.1, ion channels, hERG, SAR, antiproliferative activity Full text (file, 869,51 KB) This document has more files! More... |
3. Structure-function studies of sponge-derived compounds on the cardiac CaV3.1 channelAnne-Sophie Depuydt, Piyush A. Patel, Žan Toplak, Chinmaya Bhat, Manuela Voráčová, Irene Eteläinen, Fiammetta Vitulano, Nives Hribernik, Tihomir Tomašič, Lucija Peterlin-Mašič, 2023, original scientific article Keywords: T-type calcium channels, ion channels, purpurealidin I, bromotyrosines, marine-derived bioactive compounds Full text (file, 4,30 MB) This document has more files! More... |
4. Design of new potent and selective thiophene-based K$_V$1.3 inhibitors and their potential for anticancer activityŠpela Gubič, Žan Toplak, Štefan Možina, Tihomir Tomašič, Lucija Peterlin-Mašič, 2022, original scientific article Keywords: K$_V$1.3, potassium ion channels, antiproliferative activity, apoptosis, anticancer drugs Full text (file, 10,07 MB) This document has more files! More... |
5. Cellular excitability and ns-pulsed electric fieldsLea Rems, Aurianne Rainot, Daniel Wiczew, Natalia Szulc, Mounir Tarek, 2024, original scientific article Keywords: cell membrane, electroporation, lipid oxidation, molecular dynamics simulations, Hodgkin-Huxley models, voltage-gated ion channels Full text (file, 2,85 MB) This document has more files! More... |