31. Exploring the 5-substituted 2-aminobenzothiazole-based DNA gyrase B inhibitors active against ESKAPE pathogensMaša Sterle, Martina Durcik, Danijel Kikelj, Nace Zidar, Lucija Peterlin-Mašič, Janez Ilaš, Tihomir Tomašič, Andrej Emanuel Cotman, Anamarija Zega, 2023, original scientific article Keywords: bacteria, genetics, inhibitors, organic acids, peptides, proteins Full text (file, 4,52 MB) This document has more files! More... |
32. Exploring the interaction of N-(benzothiazol-2-yl)pyrrolamide DNA gyrase inhibitors with the GyrB ATP-binding site lipophilic floorNace Zidar, Andrej Emanuel Cotman, Wessel Sinnige, Ondřej Benek, Michaela Barančokova, Anamarija Zega, Lucija Peterlin-Mašič, Tihomir Tomašič, Janez Ilaš, Ricardo D. Enriz, Danijel Kikelj, 2024, original scientific article Keywords: antibacterial agent, DNA gyrase, ATP-binding site, N-(benzothiazol-2-yl)pyrrolamide, inhibitor, QTAIM analysis Full text (file, 2,64 MB) This document has more files! More... |
33. Identification of a novel structural class of H$_v$1 inhibitors by structure-based virtual screeningMartina Piga, Zoltán Varga, Ádám Fehér, Ferenc Papp, Eva Korpos Pintye-Gyuri, Kavya C. Bangera, Rok Frlan, Janez Ilaš, Jaka Dernovšek, Tihomir Tomašič, Nace Zidar, 2024, original scientific article Keywords: cancer, cells, inhibition, inhibitors, screening assays Full text (file, 3,20 MB) This document has more files! More... |
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