1. Fine tuning of cholinesterase and glutathione-S-transferase activities by organoruthenium(II) complexesTomaž Trobec, Kristina Sepčić, Monika C. Žužek, Jerneja Kladnik, Nina Podjed, Catarina Cardoso Páscoa, Iztok Turel, Robert Frangež, 2021, original scientific article Keywords: cholinesterase, enzyme inhibition, glutathione S-transferase, organoruthenium complex, pyrithione, β-diketone, carbonyl, glutathione transferase Full text (file, 751,83 KB) This document has more files! More... |
2. New insights into the effects of organometallic ruthenium complexes on nicotinic acetylcholine receptorsTomaž Trobec, Nicolas Lamassiaude, Evelyne Benoit, Monika C. Žužek, Kristina Sepčić, Jerneja Kladnik, Iztok Turel, Rómulo Aráoz, Robert Frangež, 2024, original scientific article Keywords: organometallic ruthenium complexes, nicotinic acetylcholine receptors, nicotinic antagonists, electrophysiology, two-electrode voltage-clamp technique Full text (file, 3,26 MB) This document has more files! More... |
3. Effects of bioinsecticidal aegerolysin-based cytolytic complexes on non-target organismsAnastasija Panevska, Gordana Glavan, Anita Jemec Kokalj, Veronika Kukuljan, Tomaž Trobec, Monika C. Žužek, Milka Vrecl, Damjana Drobne, Robert Frangež, Kristina Sepčić, 2021, original scientific article Keywords: adverse effects, aegerolysins, Apis mellifera, bioinsecticides, erylysin A, MACPF protein, non-target organisms, oyster mushroom, Porcellio scaber, toxicity Full text (file, 24,84 MB) This document has more files! More... |
4. Novel organoruthenium(II) complex C1 selectively inhibits butyrylcholinesterase without side effects on neuromuscular transmissionTomaž Trobec, Monika C. Žužek, Kristina Sepčić, Jerneja Kladnik, Iztok Turel, Robert Frangež, 2023, original scientific article Keywords: organoruthenium(II) complex, acetylcholinesterase, butyrylcholinesterase, mouse neuromuscular system, ruthenium, Alzheimer disease, neurodegenerative diseases Full text (file, 3,74 MB) This document has more files! More... |
5. Structural and functional characterization of an organometallic ruthenium complex as a potential myorelaxant drugTomaž Trobec, Monika C. Žužek, Kristina Sepčić, Jerneja Kladnik, Jakob Kljun, Iztok Turel, Evelyne Benoit, Robert Frangež, 2020, original scientific article Keywords: organoruthenium nitrophenanthroline complex, acetylcholinesterase, butyrylcholinesterase, glutathione S-transferase, mouse neuromuscular system, ruthenium, muscle relaxation, physiology, glutathione transferase Full text (file, 1,45 MB) This document has more files! More... |
6. Using virtual AChE homology screening to identify small molecules with the ability to inhibit marine biofoulingHomayon John Arabshahi, Tomaž Trobec, Valentin Foulon, Claire Hellio, Robert Frangež, Kristina Sepčić, Patrick Cahill, Johan Svenson, 2021, original scientific article Keywords: homology screening, in silico screening, in vitro enzymatic studies, cholinesterase, AChE inhibitor, antifouling Full text (file, 2,67 MB) This document has more files! More... |
7. Spatial distribution and stability of cholinesterase inhibitory protoberberine alkaloids from Papaver setiferumNeda Safa, Tomaž Trobec, Darren C. Holland, Blazej Slazak, Erik Jacobsson, Jeffrey A. Hawkes, Robert Frangež, Kristina Sepčić, Ulf Göransson, Lindon W. K. Moodie, Luke P. Robertson, 2022, original scientific article Keywords: Cholinesterase Inhibitors, Papaver, Alkaloids Full text (file, 6,46 MB) This document has more files! More... |
8. Alzheimerjeva bolezenTomaž Trobec, Monika C. Žužek, Katarina Černe, Robert Frangež, 2022, review article Keywords: Alzheimerjeva bolezen, patofiziologija, etiologija, terapija z zdravili Full text (file, 338,47 KB) This document has more files! More... |
9. Development of potent cholinesterase inhibitors based on a marine pharmacophoreVijayaragavan Elumalai, Tomaž Trobec, Maja Grundner, Christophe Labriere, Robert Frangež, Kristina Sepčić, Jørn H. Hansen, Johan Svenson, 2022, original scientific article Keywords: Nervous System Diseases, Cholinesterase Inhibitors Full text (file, 3,53 MB) This document has more files! More... |
10. Interakcije novih rutenijevih organokovinskih kompleksov s sesalskim holinergičnim sistemomTomaž Trobec, 2022, doctoral dissertation Keywords: Rutenij-kemija, organokovinske spojine, holinesterazni inhibitorji, nikotinski receptorji, membranski potenciali, mišična kontrakcija, živčno mišični stik, motorična ploščica, elektrofiziologija, metoda vpete napetosti Full text (file, 3,11 MB) |