71. Discovery and hit-to-lead optimization of benzothiazole scaffold-based DNA gyrase inhibitors with potent activity against Acinetobacter baumannii and Pseudomonas aeruginosaAndrej Emanuel Cotman, Martina Durcik, Davide Benedetto Tiz, Federica Fulgheri, Daniela Secci, Maša Sterle, Štefan Možina, Žiga Skok, Nace Zidar, Anamarija Zega, Janez Ilaš, Lucija Peterlin-Mašič, Tihomir Tomašič, Danijel Kikelj, 2023, original scientific article Keywords: antibacterial activity, bacteria, genetics, inhibitors, solubility Full text (file, 7,98 MB) This document has more files! More... |
72. Optimisation of pyrazolo[1,5-a]pyrimidin-7(4H)-one derivatives as novel Hsp90 C-terminal domain inhibitors against Ewing sarcomaŽiva Zajec, Jaka Dernovšek, Martin Distel, Martina Gobec, Tihomir Tomašič, 2023, original scientific article Keywords: cancer, Ewing sarcoma, Hsp90, inhibitor, molecular modelling Full text (file, 3,11 MB) This document has more files! More... |
73. Refined high-content imaging-based phenotypic drug screening in zebrafish xenograftsCaterina Sturtzel, Živa Zajec, Jaka Dernovšek, Tihomir Tomašič, Sabine Taschner-Mandl, Martin Distel, 2023, original scientific article Keywords: cancer models, phenotypic screening Full text (file, 5,10 MB) This document has more files! More... |
74. New aryl and acylsulfonamides as state-dependent inhibitors of Na$_v$1.3 voltage-gated sodium channelNace Zidar, Tihomir Tomašič, Danijel Kikelj, Martina Durcik, Jan Tytgat, Steve Peigneur, Marc Rogers, Alexander Haworth, Robert W. Kirby, 2023, original scientific article Keywords: voltage-gated sodium channel, Na$_v$ channel, Na$_v$1.3, inhibitor, arylsulfonamide, acylsulfonamide Full text (file, 2,36 MB) This document has more files! More... |
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76. Immunosuppressive effects of new thiophene-based K$_V$1.3 inhibitorsŠpela Gubič, Janez Ilaš, Tihomir Tomašič, Annarosa Arcangeli, Lucija Peterlin-Mašič, 2023, original scientific article Keywords: ion channel, K$_V$1.3 inhibitor, T-lymphocyte, immunosuppressive Full text (file, 2,73 MB) This document has more files! More... |
77. Exploring the 5-substituted 2-aminobenzothiazole-based DNA gyrase B inhibitors active against ESKAPE pathogensMaša Sterle, Martina Durcik, Danijel Kikelj, Nace Zidar, Lucija Peterlin-Mašič, Janez Ilaš, Tihomir Tomašič, Andrej Emanuel Cotman, Anamarija Zega, 2023, original scientific article Keywords: bacteria, genetics, inhibitors, organic acids, peptides, proteins Full text (file, 4,52 MB) This document has more files! More... |
78. Catalytic performance of Noyori–Ikariya-type ruthenium complex with tethered syn-ULTAM ligand for the asymmetric transfer hydrogenation of ketonesSimona Hašanová, Jernej Cingl, Tihomir Tomašič, Andrej Emanuel Cotman, 2024, original scientific article Keywords: asymmetric synthesis, ruthenium, hydrogenation, alcohol Full text (file, 599,43 KB) This document has more files! More... |
79. Exploring the interaction of N-(benzothiazol-2-yl)pyrrolamide DNA gyrase inhibitors with the GyrB ATP-binding site lipophilic floorNace Zidar, Andrej Emanuel Cotman, Wessel Sinnige, Ondřej Benek, Michaela Barančokova, Anamarija Zega, Lucija Peterlin-Mašič, Tihomir Tomašič, Janez Ilaš, Ricardo D. Enriz, Danijel Kikelj, 2024, original scientific article Keywords: antibacterial agent, DNA gyrase, ATP-binding site, N-(benzothiazol-2-yl)pyrrolamide, inhibitor, QTAIM analysis Full text (file, 2,64 MB) This document has more files! More... |
80. Identification of a novel structural class of H$_v$1 inhibitors by structure-based virtual screeningMartina Piga, Zoltán Varga, Ádám Fehér, Ferenc Papp, Eva Korpos Pintye-Gyuri, Kavya C. Bangera, Rok Frlan, Janez Ilaš, Jaka Dernovšek, Tihomir Tomašič, Nace Zidar, 2024, original scientific article Keywords: cancer, cells, inhibition, inhibitors, screening assays Full text (file, 3,20 MB) This document has more files! More... |