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1. Intracellular hydrolysis of small-molecule O-linked N-acetylglucosamine transferase inhibitors differs among cells and is not required for its inhibition Elena Maria Loi, Matjaž Weiss, Stane Pajk, Martina Gobec, Tihomir Tomašič, Roland J. Pieters, Marko Anderluh, 2020, original scientific article Keywords: ester hydrolysis, inhibitor, O-GlcNAc transferase, OGT inhibitor |
2. Overview of the assays to probe O-linked β-N-acetylglucosamine transferase binding and activity Cyril Balsollier, Roland J. Pieters, Marko Anderluh, 2021, review article Keywords: OGT, GlcNAcylation, O-GlcNAc transferase, bioassay, OGT inhibitor |