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1. Accessing three-branched high-affinity cereblon ligands for molecular glue and protein degrader design Robert Kuchta, Christopher Heim, Alexander Herrmann, Samuel Maiwald, Yuen Lam Dora Ng, Izidor Sosič, Tim Keuler, Jan Krönke, Michael Gütschow, Marcus D. Hartmann, Christian Steinebach, 2023, original scientific article Keywords: the Petasis borono-Mannich reaction, Strecker synthesis, CRBN ligands |
2. Heterobifunctional ligase recruiters enable pan-degradation of inhibitor of apoptosis proteins Yuen Lam Dora Ng, Aleša Bricelj, Jacqueline A. Jansen, Arunima Murgai, Kirsten Peter, Katherine A. Donovan, Michael Gütschow, Jan Krönke, Christian Steinebach, Izidor Sosič, 2023, original scientific article Keywords: antagonists, degradation, ligands, mixtures, peptides, proteins, pharmaceutical chemistry |