1. Anthranilic acid inhibitors of undecaprenyl pyrophosphate synthase (UppS), an essential enzyme for bacterial cell wall biosynthesisMarko Jukič, Kaja Rožman, Matej Sova, Hélène Barreteau, Stanislav Gobec, 2019, original scientific article Keywords: UppS, inhibitors, cell-wall, pharmacophore model, antibacterial agents, undecaprenyl pyrophosphate synthase Full text (file, 4,42 MB) This document has more files! More... |
2. Synthesis and evaluation of N-phenylpyrrolamides as DNA gyrase B inhibitorsMartina Durcik, Päivi Tammela, Michaela Barančokova, Tihomir Tomašič, Janez Ilaš, Danijel Kikelj, Nace Zidar, 2018, original scientific article Keywords: DNA gyrase, GyrB, antibacterials, inhibitors, pyrrolamides Full text (file, 452,68 KB) This document has more files! More... |
3. Antimicrobial potencial of acinobacterial inhibotors of MurA and MurB ligases in bacterium Clostridium difficileElmedine Rustemi, 2019, master's thesis Keywords: molecular biology, cloning, Clostridium difficile, Mur ligases, actinobacterial inhibitors, protein expression, insect cells, purification, inhibitory assay Full text (file, 3,69 MB) |
4. Antimicrobial and modulatory activity of selected phytochemicals and epidemiological characteristics of antibiotic resistance in Camylobacter jejuniJasna Kovač, 2015, doctoral dissertation Keywords: Campylobacter jejuni, foodborne pathogens, antibiotic resistance, resistance modulation, plant extracts, pinocembrin, Alpinia katsumadai, essential oils, phytochemicals, alpha pinene, efflux inhibitors, adaptation response, epidemiology, MLST, gyr A typing, whole genome sequences, clonal expansion, campylobacteriosis prevalence, mathematical modelling Full text (file, 28,15 MB) |
5. DPP-4 inhibitors in the prevention/treatment of pulmonary fibrosis, heart and kidney injury caused by covid-19-a therapeutic approach of choice in type 2 diabetic patients?Andrija Smelcerović, Gordana Kocic, Mihajlo Gajic, Katarina Tomović, Vukica Djordjevic, Dobrila Stankovic-Djordjevic, Marko Anderluh, 2020, original scientific article Keywords: COVID-19, diabetes, DPP-4 inhibitors, fibrosis, multi-organ injury Full text (file, 375,34 KB) This document has more files! More... |
6. Synthesis, molecular modelling and biological evaluation of novel heterodimeric, multiple ligands targeting cholinesterases and amyloid betaMichalina Hebda, Marek Bajda, Anna Więckowska, Natalia Szałaj, Anna Pasieka, Dawid Panek, Justyna Godyń, Tomasz Wichur, Damijan Knez, Stanislav Gobec, Barbara Malawska, 2016, original scientific article Keywords: cholinesterase inhibitors, molecular modelling, β-amyloid aggregation inhibitors, Alzheimer’s disease, multi-target-directed ligands (MTDL), PAMPA-BBB assay Full text (file, 3,87 MB) This document has more files! More... |
7. Synthesis and biological evaluation of benzochromenopyrimidinones as cholinesterase inhibitors and potent antioxidant, non-hepatotoxic agents for Alzheimer's diseaseYoussef Dgachi, Oscar M. Bautista-Aguilera, Mohamed Benchekroun, Hélène Martin, Alexandre Bonet, Damijan Knez, Justyna Godyń, Barbara Malawska, Stanislav Gobec, Mourad Chioua, Jana Janockova, Ondrej Soukup, Fakher Chabchoub, José Marco-Contelles, Lhassane Ismaili, 2016, original scientific article Keywords: Alzheimer's disease, quinazolinones, multicomponent reactions, multitarget-directed ligands, antioxidants, cholinesterase inhibitors, hepatotoxicity Full text (file, 1,47 MB) This document has more files! More... |
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9. Design, synthesis, and biological evaluation of 2-(benzylamino-2-hydroxyalkyl)isoindoline-1,3-diones derivatives as potential disease-modifying multifunctional anti-Alzheimer agentsDawid Panek, Anna Więckowska, Anna Pasieka, Justyna Godyń, Jakub Jończyk, Marek Bajda, Damijan Knez, Stanislav Gobec, Barbara Malawska, 2018, original scientific article Keywords: isoindoline-1, 3-dione derivatives, cholinesterase inhibitors, BACE-1 inhibitors, Aβ-aggregation, molecular modeling, multiple anti-Alzheimer's ligands Full text (file, 6,29 MB) This document has more files! More... |
10. Early Lyme borreliosis in patients treated with tumour necrosis factor-alfa inhibitorsVera Maraspin-Čarman, Petra Bogovič, Tereza Rojko, Katarina Ogrinc, Eva Ružić-Sabljić, Franc Strle, 2019, original scientific article Keywords: Lyme borreliosis, immunocompromised host, TNF-α inhibitors, erythema migrans, treatment, outcome Full text (file, 234,57 KB) This document has more files! More... |