91. Half-sandwich Ir(III) and Os(II) complexes of pyridyl-mesoionic carbenes as potential anticancer agentsJuran Kralj, Aljoša Bolje, Darija Stupin Polančec, Ivana Steiner, Tena Gržan, Ana Tupek, Nikolina Stojanović, Stephan Hohloch, Damijana Urankar, Maja Osmak, Biprajit Sarkar, Anamaria Brozović, Janez Košmrlj, 2019, original scientific article Keywords: pyridyl-mesoionic carbenes, anticancer agents, iridium, osmium Full text (outside link) |
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94. New dual inhibitors of bacterial topoisomerases with broad-spectrum antibacterial activity and in vivo efficacy against vancomycin-intermediate Staphylococcus aureusMartina Durcik, Andrej Emanuel Cotman, Žan Toplak, Štefan Možina, Žiga Skok, Maria Vittoria Piras, Nace Zidar, Janez Ilaš, Anamarija Zega, Jurij Trontelj, Danijel Kikelj, Tihomir Tomašič, Lucija Peterlin-Mašič, 2023, original scientific article Keywords: antibacterial activity, bacteria, inhibitors, genetics, inhibition, peptides and proteins Full text (file, 4,53 MB) This document has more files! More... |
95. Discovery of K$_V$1.3 ion channel inhibitorsŠpela Gubič, Louise Antonia Hendrickx, Žan Toplak, Maša Sterle, Steve Peigneur, Tihomir Tomašič, Luis A. Pardo, Jan Tytgat, Anamarija Zega, Lucija Peterlin-Mašič, 2021, review article Keywords: K$_V$1.3 channel, design of K$_V$1.3 inhibitors, mitochondrial K$_V$1.3, peptide inhibitors, small-molecule inhibitors Full text (file, 6,21 MB) This document has more files! More... |
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97. Hybrid inhibitors of DNA gyrase A and BMartina Durcik, Žiga Skok, Janez Ilaš, Nace Zidar, Anamarija Zega, Petra Szili, Gábor Draskovits, T. Revesz, Danijel Kikelj, Ákos Nyerges, Csaba Pál, Lucija Peterlin-Mašič, Tihomir Tomašič, 2021, original scientific article Keywords: antibacterial, ciprofloxacin, DNA gyrase, dual inhibitor, hybrid Full text (file, 3,42 MB) This document has more files! More... |
98. ATP-competitive inhibitors of human DNA topoisomerase IIα with improved antiproliferative activity based on N-phenylpyrrolamide scaffoldŽiga Skok, Martina Durcik, Živa Zajec, Darja Gramec, Krištof Bozovičar, Anja Pišlar, Tihomir Tomašič, Anamarija Zega, Lucija Peterlin-Mašič, Danijel Kikelj, Nace Zidar, Janez Ilaš, 2023, original scientific article Keywords: anticancer drugs, ATP-competitive inhibitors, catalytic inhibitor, cytotoxicity, human DNA topoisomerase II Full text (file, 2,83 MB) This document has more files! More... |
99. Načrtovanje zaviralcev katepsina K in avtolizina s pomočjo pristopov kemometrije in strukturno podprtega načrtovanjaJure Borišek, 2015, doctoral dissertation Keywords: farmacevtska kemija, katepsin K, avtolizin E, zaviralci, balicatib, vrednotenje, načrtovanje, kemijska struktura, klinične raziskave, neželeni učinki, lizosomotropizem, osteoporoza, zdravljenje, kemometrija, disertacije Full text (file, 4,71 MB) |
100. Napovedovanje antioksidativne aktivnosti in transmembranskega transporta derivatov pulvinske kisline in kumarinaRok Martinčič, 2015, doctoral dissertation Keywords: antioksidanti, pulvinska kislina, kumarin, derivati, antioksidativna aktivnost, transmembranski transport, bilitranslokaza, računalniško modeliranje, disertacije Full text (file, 4,69 MB) |