21. The free energy folding penalty accompanying binding of intrinsically disordered α-helical motifsSan Hadži, Jurij Lah, 2022, izvirni znanstveni članek Ključne besede: binding motif, folding penalty, folding-upon-binding, fuzziness, intrinsically disordered proteins, peptide inhibitor, pre-folding Celotno besedilo (datoteka, 1,78 MB) Gradivo ima več datotek! Več... |
22. Potent DNA gyrase inhibitors bind asymmetrically to their target using symmetrical bifurcated halogen bondsAnja Kolarič, Thomas Germe, Martina Hrast, Clare E. M. Stevenson, David M. Lawson, Nicolas P. Burton, Judit Vörös, Anthony Maxwell, Nikola Minovski, Marko Anderluh, 2021, izvirni znanstveni članek Ključne besede: antibacterials, DNA gyrase inhibitors, drug discovery, Staphylococcus aureus, intercalators, novel bacterial topoisomerase inhibitors, NBTIs, symmetrical bifurcated halogen bonds, crystal structure, novel NBTIs mechanism of action, antimicrobials, DNA-binding proteins, drug development, X-ray crystallography Celotno besedilo (datoteka, 2,00 MB) Gradivo ima več datotek! Več... |
23. Combining cross-coupling reaction and Knoevenagel condensation in the synthesis of glyco-BODIPY probes for DC-SIGN super-resolution bioimagingGiacomo Biagiotti, Edvin Purić, Iztok Urbančič, Ana Krišelj, Matjaž Weiss, Janez Mravljak, Cristina Gellini, Luigi Lay, Fabrizio Chiodo, Marko Anderluh, 2021, izvirni znanstveni članek Ključne besede: BODIPY, mannose binding lectins, stimulated emission depletion microscopy, DC-SIGN, glycan Celotno besedilo (datoteka, 4,75 MB) Gradivo ima več datotek! Več... |
24. Development of in silico classification models for binding affinity to the glucocorticoid receptorMark Stanojević, Marjan Vračko, Marija Sollner Dolenc, 2023, izvirni znanstveni članek Ključne besede: endocrine disruptions, binding to glucocorticoid receptor, in silico classification, counterpropagation artificial neural networks, DRAGON descriptors Celotno besedilo (datoteka, 2,95 MB) Gradivo ima več datotek! Več... |
25. Binding-induced diversity of a human telomeric G-quadruplex stability phase spaceDomen Oblak, San Hadži, Črtomir Podlipnik, Jurij Lah, 2022, izvirni znanstveni članek Ključne besede: G-quadruplex, G-quadruplex stability, G-quadruplex ligand binding, G-quadruplex structure, thermodynamics, DSC, human telomere repeat Celotno besedilo (datoteka, 18,01 MB) Gradivo ima več datotek! Več... |
26. CAT-SiteŽan Hafner Petrovski, Barbara Hribar-Lee, Zoran Bosnić, 2022, izvirni znanstveni članek Ključne besede: protein binding site prediction, ligands, molecular docking, machine learning, convolutional neural network Celotno besedilo (datoteka, 10,33 MB) Gradivo ima več datotek! Več... |
27. Leucine motifs stabilize residual helical structure in disordered proteinsUroš Zavrtanik, Tadej Medved, Samo Purič, Wim F. Vranken, Jurij Lah, San Hadži, 2024, izvirni znanstveni članek Ključne besede: intrinsically disordered proteins, folding-upon-binding, pre-folding, preotein recognition motif, leucine recognition motif Celotno besedilo (datoteka, 1,65 MB) Gradivo ima več datotek! Več... |