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24. The synthesis of (2R)-aziridine-2-carboxylic acid containing dipeptidesSamo Kuzmič, Martina Hrast, Rok Frlan, 2022, original scientific article Keywords: dipeptides, aziridines, biomarkers, warheads, antibacterial agents Full text (file, 406,86 KB) This document has more files! More... |
25. Discovery of a fragment hit compound targeting D-Ala:D-Ala ligase of bacterial peptidoglycan biosynthesisMatic Proj, Martina Hrast, Gregor Bajc, Rok Frlan, Anže Meden, Matej Butala, Stanislav Gobec, 2023, original scientific article Keywords: fragment-based drug discovery, hit triage, inhibitors, antibacterial agents Full text (file, 1,79 MB) This document has more files! More... |
26. Fragment-sized thiazoles in fragment-based drug discovery campaignsMatic Proj, Martina Hrast, Damijan Knez, Krištof Bozovičar, Katarina Grabrijan, Anže Meden, Stanislav Gobec, Rok Frlan, 2022, original scientific article Keywords: thiazoles, hit profiling, promiscuous compounds, frequent hitters, privileged scaffolds, fragments Full text (file, 2,30 MB) This document has more files! More... |
27. Mur ligase F as a new target for the flavonoids quercitrin, myricetin, and (–)-epicatechinMartina Hrast, Irena Zdovc, Nina Kočevar Glavač, Stanislav Gobec, Rok Frlan, 2023, original scientific article Keywords: MurF, quercitrin, myricetin, (–)-epicatechin, antibacterial activity Full text (file, 1,43 MB) This document has more files! More... |
28. Inhibition of MurA enzyme from Escherichia coli by flavonoids and their synthetic analoguesRok Frlan, Martina Hrast, Stanislav Gobec, 2023, original scientific article Keywords: assays, flavonoids, inhibition, inhibitors, peptides, proteins Full text (file, 2,97 MB) This document has more files! More... |
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30. Načrtovanje in sinteza N-(2-aminoetil)- 2,4-dihidroksibenzamidnih zaviralcev D-alanil-D-alanin ligazeGorazd Zupan, 2020, master's thesis/paper Keywords: D-alanil-D-alanin ligaza, bakterijska odpornost, nove protibakterijske učinkovine, celična stena, N-(2-aminoetil)-2, 4-dihidroksibenzamid Full text (file, 1,42 MB) |