31. Biopharmaceutical classification of desloratadine - not all drugs are classified the easy wayKatja Berginc, Nadica Sibinovska, Simon Žakelj, Jurij Trontelj, Igor Legen, 2020, izvirni znanstveni članek Ključne besede: desloratadine, BCS-based bio-waiver, luminal stability, permeability, dissolution Celotno besedilo (datoteka, 433,79 KB) Gradivo ima več datotek! Več... |
32. Stereoselective activity of 1-propargyl-4-styrylpiperidine-like analogues that can discriminate between monoamine oxidase isoforms A and BDamijan Knez, Natalia Colettis, Luca G. Iacovino, Matej Sova, Anja Pišlar, Janez Konc, Samo Lešnik, Josefina Higgs, Fabiola Kamecki, Irene Mangialavori, Ana Dolšak, Simon Žakelj, Jurij Trontelj, Janko Kos, Claudia Binda, Nora Marder Mariel, Stanislav Gobec, 2020, izvirni znanstveni članek Ključne besede: binding energy, ethyl groups, inhibition, inhibitors, molecular structure Celotno besedilo (datoteka, 6,41 MB) Gradivo ima več datotek! Več... |
33. Proof-of-concept for a miniaturized shake-flask biopharmaceutical solubility determination by sonic mixingArdita Veseli, Albin Kristl, Simon Žakelj, 2020, izvirni znanstveni članek Ključne besede: pharmacokinetics, physiologically based pharmacokinetic (PBPK) modeling gastro plus modeling, clinical trial simulation(s), bioequivalence, biopharmaceutics classification system (BCS), virtual bioequivalence (VBE) Celotno besedilo (datoteka, 565,27 KB) Gradivo ima več datotek! Več... |
34. 8-Hydroxyquinolylnitrones as multifunctional ligands for the therapy of neurodegenerative diseasesDamijan Knez, Anže Meden, Anja Pišlar, Janko Kos, Simon Žakelj, Jure Stojan, Stanislav Gobec, José Marco-Contelles, 2023, izvirni znanstveni članek Ključne besede: quinolylnitrone, butyrylcholinesterase, monoamine oxidase B, Alzheimer's disease, multifunctional ligands, 6-hydroxydopamine model, passive avoidance task, novel object recognition Celotno besedilo (datoteka, 3,96 MB) Gradivo ima več datotek! Več... |
35. How azide ion/hydrazoic acid passes through biological membranesSimona Lojevec Hartl, Simon Žakelj, Marija Sollner Dolenc, Vladimir Smrkolj, Janez Mavri, 2023, izvirni znanstveni članek Ključne besede: azide ion, hydrazoic acid, octanol/water partition coefficient, effective permeability, PAMPA, diffusion, inhibition, cytochrome c oxidase complex IV Celotno besedilo (datoteka, 985,33 KB) Gradivo ima več datotek! Več... |
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