271. Small and simple, yet sturdyKrištof Bozovičar, Tomaž Bratkovič, 2021, review article Keywords: constrained peptides, macrocycles, crosslinking, enzymatic cyclization, stapling, hairpin loop Full text (file, 2,46 MB) This document has more files! More... |
272. Extracellular cystatin F is internalised by cytotoxic T lymphocytes and decreases their cytotoxicityMateja Prunk, Milica Perišić, Tanja Jakoš, Jerica Sabotič, Urban Švajger, Janko Kos, 2020, original scientific article Keywords: cystatin F, cathepsins, cytotoxic lymphocytes, granzymes, perforin, TALL-104 Full text (file, 3,56 MB) This document has more files! More... |
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274. Hybrid inhibitors of DNA gyrase A and BMartina Durcik, Žiga Skok, Janez Ilaš, Nace Zidar, Anamarija Zega, Petra Szili, Gábor Draskovits, T. Revesz, Danijel Kikelj, Ákos Nyerges, Csaba Pál, Lucija Peterlin-Mašič, Tihomir Tomašič, 2021, original scientific article Keywords: antibacterial, ciprofloxacin, DNA gyrase, dual inhibitor, hybrid Full text (file, 3,42 MB) This document has more files! More... |
275. Vaccinomics and adversomics in the era of precision medicineJasna Omersel, Nataša Karas Kuželički, 2020, review article Keywords: adversomics, COVID-19, genetics, hepatitis B, human Papilloma virus, MMR vaccine, precision medicine, vaccinomics Full text (file, 1,21 MB) This document has more files! More... |
276. Bromo-cyclobutenaminones as new covalent UDP-N-acetylglucosamine enolpyruvyl transferase (MurA) inhibitorsDavid J. Hamilton, Péter Ábrányi-Balogh, Aaron Keeley, László Petri, Martina Hrast, Tímea Imre, Maikel Wijtmans, Stanislav Gobec, Iwan J. P. de Esch, György Keserü M., 2020, original scientific article Keywords: covalent inhibitor, MurA, cyclobutenaminone, antibacterial, irreversible Full text (file, 1,08 MB) This document has more files! More... |
277. Synthesis of conformationally constrained D-Glu-meso-DAP analogs as innate immune agonistsSamo Guzelj, Žiga Jakopin, 2020, original scientific article Keywords: NOD1 agonist, constrained meso-DAP mimetics, NOD1 activation, innate immune agonist, bioisosteric replacement, rigidization Full text (file, 1,65 MB) This document has more files! More... |
278. Echinacea angustifolia DC. lipophilic extract patch for skin applicationDritan Hasa, Simon Žakelj, Iztok Grabnar, Francesco Cilurzo, Stefano Dall'Acqua, Antonella Riva, Beatrice Perissutti, Dario Voinovich, 2020, original scientific article Keywords: Echinacea angustifolia lipophilic extract, tetraene, drug-in-adhesive patch, in vitro skin permeation, pharmacokinetics Full text (file, 1,40 MB) This document has more files! More... |
279. Discovery of novel Hsp90 C-terminal inhibitors using 3D-pharmacophores derived from molecular dynamics simulationsTihomir Tomašič, Martina Durcik, Bradley M. Keegan, Darja Gramec, Živa Zajec, Brian S. J. Blagg, Sharon D. Bryant, 2020, original scientific article Keywords: allosteric, cancer, Hsp90, inhibitor, molecular dynamics, pharmacophores, virtual screening Full text (file, 7,84 MB) This document has more files! More... |
280. Silver fir (Abies alba L.) polyphenolic extract shows beneficial influence on chondrogenesis in vitro under normal and inflammatory conditionsMateja Sirše, Samo K. Fokter, Borut Štrukelj, Janja Zupan, 2020, original scientific article Keywords: mesenchymal stem cells, mesenchymal stromal cells, polyphenols, chondrogenesis, inflammation, subchondral bone, osteoarthritis Full text (file, 3,24 MB) This document has more files! More... |