131. Discovery of a fragment hit compound targeting D-Ala:D-Ala ligase of bacterial peptidoglycan biosynthesisMatic Proj, Martina Hrast, Gregor Bajc, Rok Frlan, Anže Meden, Matej Butala, Stanislav Gobec, 2023, original scientific article Keywords: fragment-based drug discovery, hit triage, inhibitors, antibacterial agents Full text (file, 1,79 MB) This document has more files! More... |
132. Next-generation heterocyclic electrophiles as small-molecule covalent MurA inhibitorsPéter Ábrányi-Balogh, Aaron Keeley, György G. Ferenczy, László Petri, Tímea Imre, Katarina Grabrijan, Martina Hrast, Damijan Knez, Janez Ilaš, Stanislav Gobec, György Keserü M., 2022, original scientific article Keywords: covalent inhibitor, heterocyclic electrophiles, cysteine labelling, quaternization, MurA Full text (file, 1,46 MB) This document has more files! More... |
133. Dietary iron intake and biomarkers of iron status in Slovenian populationŽiva Lavriša, Hristo Hristov, Maša Hribar, Barbara Koroušić-Seljak, Matej Gregorič, Urška Blaznik, Katja Zaletel, Adrijana Oblak, Joško Osredkar, Anita Kušar, Katja Žmitek, Mitja Lainščak, Igor Pravst, 2022, original scientific article Keywords: iron, intake, ferritin, haemoglobin, deficiency, Slovenia, EU Menu, Nutrihealth Full text (file, 1,71 MB) This document has more files! More... |
134. The synthesis of (2R)-aziridine-2-carboxylic acid containing dipeptidesSamo Kuzmič, Martina Hrast, Rok Frlan, 2022, original scientific article Keywords: dipeptides, aziridines, biomarkers, warheads, antibacterial agents Full text (file, 406,86 KB) This document has more files! More... |
135. Characterization of the spray droplets and spray pattern by means of innovative optical microscopy measurement method with the high-speed cameraNejc Koračin, Matevž Zupančič, Franc Vrečer, Grega Hudovornik, Iztok Golobič, 2022, original scientific article Keywords: film coating, atomization process, image processing, microscopy, high-speed image acquisition, pharmaceutics Full text (file, 4,50 MB) This document has more files! More... |
136. Association of Zn and Cu levels in cord blood and maternal milk with pregnancy outcomes among the Slovenian populationJoško Osredkar, Živa Miriam Geršak, Nataša Karas Kuželički, Janja Snoj Tratnik, Darja Mazej, Ingrid Falnoga, Milena Horvat, Ksenija Geršak, 2022, original scientific article Keywords: cord blood, maternal milk, gestational age, birth weight Full text (file, 1,38 MB) This document has more files! More... |
137. N-hydroxy-N-propargylamide derivatives of ferulic acidOscar M. Bautista-Aguilera, José M. Alonso, Marco Catto, Isabel Iriepa, Damijan Knez, Stanislav Gobec, José Marco-Contelles, 2022, original scientific article Keywords: cholinesterases, ferulic acid, molecular modelling, monoamine oxidase, radical-scavenger, antioxidant Full text (file, 792,16 KB) This document has more files! More... |
138. Comparison of the robustness of pellet film coating with and without in-process coating thickness evaluationTeja Brezovar, Sandi Svetič, Rok Dreu, 2022, original scientific article Keywords: pellets, coating of pellets, prolonged release coating, PAT, image analysis, residual water Full text (file, 1,29 MB) This document has more files! More... |
139. Evaluation of novel cathepsin-X inhibitors in vitro and in vivo and their ability to improve cathepsin-B-directed antitumor therapyAna Mitrović, Janja Završnik, Georgy Mikhaylov, Damijan Knez, Urša Pečar Fonović, Petra Matjan-Štefin, Miha Butinar, Stanislav Gobec, Boris Turk, Janko Kos, 2022, original scientific article Keywords: cathepsin X, cathepsin B, inhibitors, cancer, antitumor therapy, invasion Full text (file, 8,24 MB) This document has more files! More... |
140. Catalytic stereoconvergent synthesis of homochiral β‑CF$_3$, β‑SCF$_3$, and β‑OCF$_3$ benzylic alcoholsAndrej Emanuel Cotman, Pavel A. Dub, Maša Sterle, Matic Lozinšek, Jaka Dernovšek, Živa Zajec, Anamarija Zega, Tihomir Tomašič, Dominique Cahard, 2022, original scientific article Keywords: adaptive crystals, asymmetric catalysis, density functional calculations, drug design, fluorine, hydrogenation, kinetic resolution, ruthenium, alcohols, catalysts, crystals, ketones, stereoselectivity Full text (file, 2,08 MB) This document has more files! More... |