11. Novel selective IDO1 inhibitors with isoxazolo[5,4-d]pyrimidin-4(5H)-one scaffoldAna Dolšak, Tomaž Bratkovič, Larisa Mlinarič, Eva Ogorevc, Urban Švajger, Stanislav Gobec, Matej Sova, 2021, original scientific article Keywords: indoleamine 2, 3-dioxygenase 1, selective inhibitors, isoxazolo[5, 4-d]pyrimidin-4(5H)-one, immunomodulation, cancer Full text (file, 19,67 MB) This document has more files! More... |
12. Drug delivery strategies for curcumin and other natural Nrf2 modulators of oxidative stress-related diseasesNina Katarina Grilc, Matej Sova, Julijana Kristl, 2021, review article Keywords: Nrf2 modulator, oxidative stress, oral bioavailability, poor solubility, curcumin, resveratrol, solid dispersions, SMEDDS, nanoparticles, micelles Full text (file, 2,60 MB) This document has more files! More... |
13. Nanotechnology-based drug delivery to improve the therapeutic benefits of NRF2 modulators in cancer therapyZerrin Sezgin-Bayindir, Sonia Losada-Barreiro, Carlos Bravo-Díaz, Matej Sova, Julijana Kristl, Luciano Saso, 2021, review article Keywords: NRF2 modulators, anticancer agents, nanoparticles, drug delivery, drug targeting Full text (file, 1,96 MB) This document has more files! More... |
14. Strukturno podprto načrtovanje, sinteza in vrednotenje novih zaviralcev indolamin 2,3-dioksigenaze in modulatorjev toll-u podobnih receptorjev tipa 7 in 8Ana Dolšak, 2021, doctoral dissertation Keywords: Toll-u podoben receptor 7, Toll-u podoben receptor 8, negativni modulator TLR8, virtualno rešetanje, tvorba C-C vezi, Suzuki reakcija, substituirani pirimidi, imunski sistem, farmacevtska kemija
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15. Strukturno-podprto načrtovanje, sinteza in vrednotenje novih zaviralcev biosinteze peptidoglikanaKaja Rožman, 2018, doctoral dissertation Keywords: bakterijske infekcije, zdravljenje, protibakterijske učinkovine, celična stena, peptidoglikan, biosinteza, encimi, encimi Mur, undekaprelin pirofosfat sintetaza, penicilin vezoči protein 2a, encimski inhibitorji, mikobakterije, mikolne kisline, načrtovanje, sinteza, vrednotenje, rešetanje, disertacije Full text (file, 8,64 MB) |
16. 4-phenethyl-1-propargylpiperidine-derived dual inhibitors of butyrylcholinesterase and monoamine oxidase BTjaša Mazej, Damijan Knez, Anže Meden, Stanislav Gobec, Matej Sova, 2021, original scientific article Keywords: Alzheimer's disease, butyrylcholinesterase, monoamine oxidase B, inhibitors, multi-target-directed ligands, multifunctional ligands Full text (file, 3,88 MB) This document has more files! More... |
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