61. Stereoselective activity of 1-propargyl-4-styrylpiperidine-like analogues that can discriminate between monoamine oxidase isoforms A and BDamijan Knez, Natalia Colettis, Luca G. Iacovino, Matej Sova, Anja Pišlar, Janez Konc, Samo Lešnik, Josefina Higgs, Fabiola Kamecki, Irene Mangialavori, Ana Dolšak, Simon Žakelj, Jurij Trontelj, Janko Kos, Claudia Binda, Nora Marder Mariel, Stanislav Gobec, 2020, izvirni znanstveni članek Ključne besede: binding energy, ethyl groups, inhibition, inhibitors, molecular structure Celotno besedilo (datoteka, 6,41 MB) Gradivo ima več datotek! Več... |
62. Semisynthetic teicoplanin derivatives with dual antimicrobial activity against SARS-CoV-2 and multiresistant bacteriaIlona Bereczki, Vladimir Vimberg, Eszter Lőrincz, Henrietta Papp, Lajos Nagy, Sándor Kéki, Gyula Batta, Ana Mitrović, Janko Kos, Áron Zsigmond, 2022, izvirni znanstveni članek Celotno besedilo (datoteka, 1,83 MB) Gradivo ima več datotek! Več... |
63. Evaluation of novel cathepsin-X inhibitors in vitro and in vivo and their ability to improve cathepsin-B-directed antitumor therapyAna Mitrović, Janja Završnik, Georgy Mikhaylov, Damijan Knez, Urša Pečar Fonović, Petra Matjan-Štefin, Miha Butinar, Stanislav Gobec, Boris Turk, Janko Kos, 2022, izvirni znanstveni članek Ključne besede: cathepsin X, cathepsin B, inhibitors, cancer, antitumor therapy, invasion Celotno besedilo (datoteka, 8,24 MB) Gradivo ima več datotek! Več... |
64. 8-Hydroxyquinolylnitrones as multifunctional ligands for the therapy of neurodegenerative diseasesDamijan Knez, Anže Meden, Anja Pišlar, Janko Kos, Simon Žakelj, Jure Stojan, Stanislav Gobec, José Marco-Contelles, 2023, izvirni znanstveni članek Ključne besede: quinolylnitrone, butyrylcholinesterase, monoamine oxidase B, Alzheimer's disease, multifunctional ligands, 6-hydroxydopamine model, passive avoidance task, novel object recognition Celotno besedilo (datoteka, 3,96 MB) Gradivo ima več datotek! Več... |
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