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43. Načrtovanje in sinteza benzotiazolnih zaviralcev HSP90 in DNA-girazeAmadeja Zgaga, 2017, master's thesis Keywords: DNA giraze, Hsp90, protibakterijsko delovanje, protivirusno delovanje, sintezni postopki, topoizomeraza tip II, bakterijska rezistenca Full text (file, 1,53 MB) |
44. Načrtovanje in sinteza C-manozidov in N-manodizov kot potencialnih antagonistov lektina FimHNina Malešič, 2017, master's thesis Keywords: bakterijske okužbe, antiadhezivna terapija, protimikrobne učinkovine, Escherichia coli, alfa-D-manoza, C-manozidi, N-manozidi, lektin FimH, bakterije Full text (outside link) |
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47. Novel scaffolds for modulation of NOD2 identified by pharmacophore-based virtual screeningSamo Guzelj, Tihomir Tomašič, Žiga Jakopin, 2022, original scientific article Keywords: antagonist, homology modeling, NOD2, Nucleotide-binding oligomerization, pharmacophore modeling, virtual screening Full text (file, 24,71 MB) This document has more files! More... |
48. Discovery of a new drug-like series of OGT inhibitors by virtual screeningElena Maria Loi, Tihomir Tomašič, Cyril Balsollier, Kevin van Eekelen, Matjaž Weiss, Martina Gobec, Matthew G Alteen, David J. Vocadlo, Roland J. Pieters, Marko Anderluh, 2022, original scientific article Keywords: O-GlcNAc transferase, OGT inhibitors, virtual screening, pharmaceutical chemistry Full text (file, 10,66 MB) This document has more files! More... |
49. Discovery of substituted oxadiazoles as a novel scaffold for DNA gyrase inhibitorsŽiga Jakopin, Janez Ilaš, Michaela Barančokova, Matjaž Brvar, Päivi Tammela, Marija Sollner Dolenc, Tihomir Tomašič, Danijel Kikelj, 2017, original scientific article Keywords: 1, 2, 4-oxadiazoles, DNA gyrase inhibition, topoisomerase IV inhibition, antibacterial screening, computer-aided drug design Full text (file, 1,45 MB) This document has more files! More... |
50. Design, synthesis and biological evaluation of 4,5-dibromo-N-(thiazol-2-yl)-1H-pyrrole-2-carboxamide derivatives as novel DNA gyrase inhibitorsTihomir Tomašič, Matic Mirt, Michaela Barančokova, Janez Ilaš, Nace Zidar, Päivi Tammela, Danijel Kikelj, 2017, original scientific article Keywords: antibacterial, DNA gyrase, docking, inhibitor, thiazole Full text (file, 1,60 MB) This document has more files! More... |