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173. Screening of big pharma’s library against various in-house biological targetsDamijan Knez, Stanislav Gobec, Martina Hrast, 2022, original scientific article Keywords: Merck Mini Library, screening, MurA, MurC, human MAO-A/B, human BChE, murine AchE Full text (file, 8,55 MB) This document has more files! More... |
174. Načrtovanje in sinteza hidroksietilaminskih inhibitorjev biosinteze peptidoglikanaMatej Sova, 2009, doctoral dissertation Keywords: bakterije, učinkovine, protibakterijske, encimi, analiza spojin, sinteza, hidroksietilamini Full text (file, 15,84 MB) |
175. Methylation of selenocysteine catalysed by thiopurine S-methyltransferaseDunja Urbančič, Anita Kotar, Alenka Šmid, Marko Jukič, Stanislav Gobec, Lars Martensson, Janez Plavec, Irena Mlinarič-Raščan, 2019, original scientific article Keywords: binding analysis, enzymatic methylation, NMR spectroscopy, S-adenosylmethionine, selenocysteine, thiopurine S-methyltransferase Full text (file, 1,48 MB) This document has more files! More... |
176. Development of potent reversible selective inhibitors of butyrylcholinesterase as fluorescent probesStane Pajk, Damijan Knez, Urban Košak, Maja Zorović, Xavier Brazzolotto, Nicolas Coquelle, Florian Nachon, Jacques-Philippe Colletier, Marko Živin, Jure Stojan, Stanislav Gobec, 2020, original scientific article Keywords: butyrylcholinesterase, inhibitor, probe, fluorescence Full text (file, 1,60 MB) This document has more files! More... |
177. Fragment-sized and bidentate (immuno)proteasome inhibitors derived from cysteine and threonine targeting warheadsLevente Kollár, Martina Gobec, Matic Proj, Lara Smrdel, Damijan Knez, Stanislav Gobec, Izidor Sosič, György Keserü M., 2021, original scientific article Keywords: immunoproteasome, benzoxazole-2-carbonitriles, bidentate covalent inhibitors, fragments, non-covalent recognition Full text (file, 1,17 MB) This document has more files! More... |
178. Treatment of canine cognitive dysfunction with novel butyrylcholinesterase inhibitorMaja Zakošek, Sonja Prpar Mihevc, Malan Štrbenc, Urban Košak, Ilija German Ilić, Jurij Trontelj, Simon Žakelj, Stanislav Gobec, Darja Pavlin, Gregor Majdič, 2021, original scientific article Keywords: Alzheimer’s disease, butyrylcholinesterase, butyrylcholinesterase inhibitor, canine cognitive dysfunction, canine dementia scale, dogs Full text (file, 1,34 MB) This document has more files! More... |
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