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4. Intracellular hydrolysis of small-molecule O-linked N-acetylglucosamine transferase inhibitors differs among cells and is not required for its inhibitionElena Maria Loi, Matjaž Weiss, Stane Pajk, Martina Gobec, Tihomir Tomašič, Roland J. Pieters, Marko Anderluh, 2020, original scientific article Keywords: ester hydrolysis, inhibitor, O-GlcNAc transferase, OGT inhibitor Full text (file, 1,90 MB) This document has more files! More... |
5. Overview of the assays to probe O-linked β-N-acetylglucosamine transferase binding and activityCyril Balsollier, Roland J. Pieters, Marko Anderluh, 2021, review article Keywords: OGT, GlcNAcylation, O-GlcNAc transferase, bioassay, OGT inhibitor Full text (file, 5,14 MB) This document has more files! More... |
6. Inhibition of O-GlcNAc transferase alters the differentiation and maturation process of human monocyte derived dendritic cellsMatjaž Weiss, Marko Anderluh, Martina Gobec, 2021, original scientific article Keywords: O-GlcNAcylation, O-GlcNAc transferase (OGT), monocyte derived DCs, OSMI-1, immunometabolism, pharmaceutical chemistry Full text (file, 2,84 MB) This document has more files! More... |
7. Discovery of a new drug-like series of OGT inhibitors by virtual screeningElena Maria Loi, Tihomir Tomašič, Cyril Balsollier, Kevin van Eekelen, Matjaž Weiss, Martina Gobec, Matthew G Alteen, David J. Vocadlo, Roland J. Pieters, Marko Anderluh, 2022, original scientific article Keywords: O-GlcNAc transferase, OGT inhibitors, virtual screening, pharmaceutical chemistry Full text (file, 10,66 MB) This document has more files! More... |
8. New quinolinone O-GlcNAc transferase inhibitors based on fragment growthMatjaž Weiss, Elena Maria Loi, Maša Sterle, Cyril Balsollier, Tihomir Tomašič, Roland J. Pieters, Martina Gobec, Marko Anderluh, 2021, original scientific article Keywords: O-GlcNAc, O-GlcNAc transferase, protein glycosylation, fragments growth, molecular docking Full text (file, 1,37 MB) This document has more files! More... |