31. Discovery of benzothiazole scaffold-based DNA gyrase B inhibitorsMarina Gjorgjieva, Tihomir Tomašič, Michaela Barančokova, Sotirios Katsamakas, Janez Ilaš, Päivi Tammela, Lucija Peterlin-Mašič, Danijel Kikelj, 2016, original scientific article Keywords: organoruthenium complexes, diketonates, anticancer drugs, ROS, cytotoxicity, cell cycle arrest Full text (file, 1,17 MB) This document has more files! More... |
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33. Synthesis, antiproliferative effect and topoisomerase II inhibitory activity of 3-methyl-2-phenyl-1H-indolesNace Zidar, Daniela Secci, Tihomir Tomašič, Lucija Peterlin-Mašič, Danijel Kikelj, Daniele Passarella, Aida Nelly Garcia Argaez, Mariafrancesca Hyeraci, Lisa Via Dalla, 2020, original scientific article Keywords: 3-Methyl-2-phenyl-1H-indole, antiproliferative activity, topoisomerase II, apoptosis Full text (file, 3,09 MB) This document has more files! More... |
34. Exploring the chemical space of benzothiazole-based DNA gyrase B inhibitorsŽiga Skok, Michaela Barančokova, Ondřej Benek, Cristina Durante Cruz, Päivi Tammela, Tihomir Tomašič, Nace Zidar, Lucija Peterlin-Mašič, Anamarija Zega, Danijel Kikelj, Janez Ilaš, 2020, original scientific article Keywords: DNA gyrase, topoisomerase IV, GyrB, ParE, antibacterial benzothiazole Full text (file, 2,22 MB) This document has more files! More... |
35. Efficient synthesis of hydroxy-substituted 2-aminobenzo[d]thiazole-6-carboxylic acid derivatives as new building blocks in drug discoveryMartina Durcik, Žan Toplak, Nace Zidar, Janez Ilaš, Anamarija Zega, Danijel Kikelj, Lucija Peterlin-Mašič, Tihomir Tomašič, 2020, original scientific article Keywords: benzo[d]thiazol, medicinal chemistry Full text (file, 1,03 MB) This document has more files! More... |
36. Rational design of balanced dual-targeting antibiotics with limited resistanceÁkos Nyerges, Tihomir Tomašič, Martina Durcik, T. Revesz, Petra Szili, Žiga Skok, Nace Zidar, Janez Ilaš, Anamarija Zega, Danijel Kikelj, Lucija Peterlin-Mašič, 2020, original scientific article Keywords: antibiotics, bacterial resistance, bacterial targets Full text (file, 2,33 MB) This document has more files! More... |
37. Discovery and hit-to-lead optimization of benzothiazole scaffold-based DNA gyrase inhibitors with potent activity against Acinetobacter baumannii and Pseudomonas aeruginosaAndrej Emanuel Cotman, Martina Durcik, Davide Benedetto Tiz, Federica Fulgheri, Daniela Secci, Maša Sterle, Štefan Možina, Žiga Skok, Nace Zidar, Anamarija Zega, Janez Ilaš, Lucija Peterlin-Mašič, Tihomir Tomašič, Danijel Kikelj, 2023, original scientific article Keywords: antibacterial activity, bacteria, genetics, inhibitors, solubility Full text (file, 7,98 MB) This document has more files! More... |
38. New aryl and acylsulfonamides as state-dependent inhibitors of Na$_v$1.3 voltage-gated sodium channelNace Zidar, Tihomir Tomašič, Danijel Kikelj, Martina Durcik, Jan Tytgat, Steve Peigneur, Marc Rogers, Alexander Haworth, Robert W. Kirby, 2023, original scientific article Keywords: voltage-gated sodium channel, Na$_v$ channel, Na$_v$1.3, inhibitor, arylsulfonamide, acylsulfonamide Full text (file, 2,36 MB) This document has more files! More... |
39. Exploring the 5-substituted 2-aminobenzothiazole-based DNA gyrase B inhibitors active against ESKAPE pathogensMaša Sterle, Martina Durcik, Danijel Kikelj, Nace Zidar, Lucija Peterlin-Mašič, Janez Ilaš, Tihomir Tomašič, Andrej Emanuel Cotman, Anamarija Zega, 2023, original scientific article Keywords: bacteria, genetics, inhibitors, organic acids, peptides, proteins Full text (file, 4,52 MB) This document has more files! More... |
40. Exploring the interaction of N-(benzothiazol-2-yl)pyrrolamide DNA gyrase inhibitors with the GyrB ATP-binding site lipophilic floorNace Zidar, Andrej Emanuel Cotman, Wessel Sinnige, Ondřej Benek, Michaela Barančokova, Anamarija Zega, Lucija Peterlin-Mašič, Tihomir Tomašič, Janez Ilaš, Ricardo D. Enriz, Danijel Kikelj, 2024, original scientific article Keywords: antibacterial agent, DNA gyrase, ATP-binding site, N-(benzothiazol-2-yl)pyrrolamide, inhibitor, QTAIM analysis Full text (file, 2,64 MB) This document has more files! More... |