11. Discovery of novel small-molecule compounds with selective cytotoxicity for Burkittʼs lymphoma cells using 3D ligand-based virtual screeningMartina Gobec, Izidor Sosič, Boris Brus, Aleš Obreza, Stanislav Gobec, Irena Mlinarič-Raščan, 2014, original scientific article Keywords: Burkittʼs lymphoma, ligand-based, similarity search, selectivity Full text (file, 1,78 MB) This document has more files! More... |
12. Synthesis of 3-amino-4-substituted monocyclic ß-lactams—important structural motifs in medicinal chemistryKatarina Grabrijan, Nika Strašek Benedik, Stanislav Gobec, 2022, original scientific article Keywords: monocyclic ß-lactam, Staudinger [2+2] cyclocondensation, cerium ammonium nitrate, hydrazine hydrate, 3-amino-4-substituted azetidin-2-one, inhibitory activities Full text (file, 3,51 MB) This document has more files! More... |
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17. Novel selective IDO1 inhibitors with isoxazolo[5,4-d]pyrimidin-4(5H)-one scaffoldAna Dolšak, Tomaž Bratkovič, Larisa Mlinarič, Eva Ogorevc, Urban Švajger, Stanislav Gobec, Matej Sova, 2021, original scientific article Keywords: indoleamine 2, 3-dioxygenase 1, selective inhibitors, isoxazolo[5, 4-d]pyrimidin-4(5H)-one, immunomodulation, cancer Full text (file, 19,67 MB) This document has more files! More... |
18. Analytical techniques for structural characterization of proteins in solid pharmaceutical formsAljoša Bolje, Stanislav Gobec, 2021, review article Keywords: solid pharmaceuticals, lyophilization, analytical tools, protein characterization, protein structure, formulation development, antibody, excipients, stable drug product, safe drug Full text (file, 7,49 MB) This document has more files! More... |
19. Design, synthesis, and biological evaluation of 2-(benzylamino-2-hydroxyalkyl)isoindoline-1,3-diones derivatives as potential disease-modifying multifunctional anti-Alzheimer agentsDawid Panek, Anna Więckowska, Anna Pasieka, Justyna Godyń, Jakub Jończyk, Marek Bajda, Damijan Knez, Stanislav Gobec, Barbara Malawska, 2018, original scientific article Keywords: isoindoline-1, 3-dione derivatives, cholinesterase inhibitors, BACE-1 inhibitors, Aβ-aggregation, molecular modeling, multiple anti-Alzheimer's ligands Full text (file, 6,29 MB) This document has more files! More... |
20. Načrtovanje, sinteza in vrednotenje potencialnih učinkovin za zdravljenje Alzheimerjeve bolezni z multiplim mehanizmom delovanjaDamijan Knez, 2017, doctoral dissertation Keywords: nevrodegenerativne bolezni, zdravila, zaviralci holin-esteraz, zdravilne učinkovine, načrtovanje, sinteza, vrednotenje, Alzheimerjeva bolezen zdravljenje, učinkovine z večvrstnim delovanjem Full text (file, 10,12 MB) |