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132. Novel selective IDO1 inhibitors with isoxazolo[5,4-d]pyrimidin-4(5H)-one scaffoldAna Dolšak, Tomaž Bratkovič, Larisa Mlinarič, Eva Ogorevc, Urban Švajger, Stanislav Gobec, Matej Sova, 2021, original scientific article Keywords: indoleamine 2, 3-dioxygenase 1, selective inhibitors, isoxazolo[5, 4-d]pyrimidin-4(5H)-one, immunomodulation, cancer Full text (file, 19,67 MB) This document has more files! More... |
133. Analytical techniques for structural characterization of proteins in solid pharmaceutical formsAljoša Bolje, Stanislav Gobec, 2021, review article Keywords: solid pharmaceuticals, lyophilization, analytical tools, protein characterization, protein structure, formulation development, antibody, excipients, stable drug product, safe drug Full text (file, 7,49 MB) This document has more files! More... |
134. Design, synthesis, and biological evaluation of 2-(benzylamino-2-hydroxyalkyl)isoindoline-1,3-diones derivatives as potential disease-modifying multifunctional anti-Alzheimer agentsDawid Panek, Anna Więckowska, Anna Pasieka, Justyna Godyń, Jakub Jończyk, Marek Bajda, Damijan Knez, Stanislav Gobec, Barbara Malawska, 2018, original scientific article Keywords: isoindoline-1, 3-dione derivatives, cholinesterase inhibitors, BACE-1 inhibitors, Aβ-aggregation, molecular modeling, multiple anti-Alzheimer's ligands Full text (file, 6,29 MB) This document has more files! More... |
135. Načrtovanje, sinteza in vrednotenje potencialnih učinkovin za zdravljenje Alzheimerjeve bolezni z multiplim mehanizmom delovanjaDamijan Knez, 2017, doctoral dissertation Keywords: nevrodegenerativne bolezni, zdravila, zaviralci holin-esteraz, zdravilne učinkovine, načrtovanje, sinteza, vrednotenje, Alzheimerjeva bolezen zdravljenje, učinkovine z večvrstnim delovanjem Full text (file, 10,12 MB) |
136. Razvoj računalniške baze bioizosternih zamenjav in programa za virtualno rešetanje na osnovi ligandaSamo Lešnik, 2017, doctoral dissertation Keywords: farmacija, načrtovanje zdravilnih učinkovin, računalniške metode, računalniško podprto načrtovanje, računalniški algoritmi, teorija grafov, knjižnice molekul, virtualno rešetanje, tarče, ligandi, bioizosterije, skeletni preskok, bioaktivne snovi, Alzheimerjeva bolezen, LiSiCa - Ligand Similarity using Clique Algorithm, LiSiCa algoritem, baza BoBER, doktorske disertacije Full text (file, 27,89 MB) |
137. Strukturno-podprto načrtovanje, sinteza in vrednotenje novih zaviralcev biosinteze peptidoglikanaKaja Rožman, 2018, doctoral dissertation Keywords: bakterijske infekcije, zdravljenje, protibakterijske učinkovine, celična stena, peptidoglikan, biosinteza, encimi, encimi Mur, undekaprelin pirofosfat sintetaza, penicilin vezoči protein 2a, encimski inhibitorji, mikobakterije, mikolne kisline, načrtovanje, sinteza, vrednotenje, rešetanje, disertacije Full text (file, 8,64 MB) |
138. Upregulation of cathepsin X in glioblastomaBernarda Majc, Anamarija Habič, Metka Novak, Ana Rotter, Andrej Porčnik, Jernej Mlakar, Vera Župunski, Urša Pečar Fonović, Damijan Knez, Nace Zidar, Stanislav Gobec, Janko Kos, Tamara Lah Turnšek, Anja Pišlar, Barbara Breznik, 2022, original scientific article Keywords: glioblastoma, cathepsin X, γ-enolase, tumor microenvironment, glioblastoma stem cells, cathepsin X inhibitors Full text (file, 3,50 MB) This document has more files! More... |
139. Synthesis and biochemical evaluation of warhead-decorated psoralens as (immuno)proteasome inhibitorsEva Shannon Schiffrer, Matic Proj, Martina Gobec, Luka Rejc, Andrej Šterman, Janez Mravljak, Stanislav Gobec, Izidor Sosič, 2021, original scientific article Keywords: immunoproteasome, psoralen core, non-peptidic, electrophilic compounds, warhead scan Full text (file, 3,29 MB) This document has more files! More... |
140. Application of the N-dibenzyl protective group in the preparation of β-lactam pseudopeptidesRok Frlan, Martina Hrast, Stanislav Gobec, 2019, original scientific article Keywords: β-lactams, dibenzylamino, Mitsunobu reaction, nocardicin, pseudopeptides Full text (file, 1,55 MB) This document has more files! More... |