61. Upregulation of cathepsin X in glioblastomaBernarda Majc, Anamarija Habič, Metka Novak, Ana Rotter, Andrej Porčnik, Jernej Mlakar, Vera Župunski, Urša Pečar Fonović, Damijan Knez, Nace Zidar, Stanislav Gobec, Janko Kos, Tamara Lah Turnšek, Anja Pišlar, Barbara Breznik, 2022, original scientific article Keywords: glioblastoma, cathepsin X, γ-enolase, tumor microenvironment, glioblastoma stem cells, cathepsin X inhibitors Full text (file, 3,50 MB) This document has more files! More... |
62. New dual inhibitors of bacterial topoisomerases with broad-spectrum antibacterial activity and in vivo efficacy against vancomycin-intermediate Staphylococcus aureusMartina Durcik, Andrej Emanuel Cotman, Žan Toplak, Štefan Možina, Žiga Skok, Maria Vittoria Piras, Nace Zidar, Janez Ilaš, Anamarija Zega, Jurij Trontelj, Danijel Kikelj, Tihomir Tomašič, Lucija Peterlin-Mašič, 2023, original scientific article Keywords: antibacterial activity, bacteria, inhibitors, genetics, inhibition, peptides and proteins Full text (file, 4,53 MB) This document has more files! More... |
63. Načrtovanje, sinteza in vrednotenje novih ATP-kompetitivnih zaviralcev človeške DNA-topoiomeraze II kot potencialnih protirakavih učinkovinŽiga Skok, 2020, doctoral dissertation Keywords: DNA-topoizomeraza II, protirakave učinkovine, funkcija topoizmeraz, testiranje zaviralne aktivnosti, sinteza zaviralcev, sintezni postopki Full text (file, 6,60 MB) |
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65. Structure-activity relationships of benzothiazole-based Hsp90 C-terminal-domain inhibitorsJaka Dernovšek, Živa Zajec, Martina Durcik, Lucija Peterlin-Mašič, Martina Gobec, Nace Zidar, Tihomir Tomašič, 2021, original scientific article Keywords: allostery, Hsp90, benzothiazole, cancer, inhibitor, cancer therapy Full text (file, 7,92 MB) This document has more files! More... |
66. Neuroinflammation-induced upregulation of glial cathepsin X expression and activity in vivoAnja Pišlar, Larisa Tratnjek, Gordana Glavan, Nace Zidar, Marko Živin, Janko Kos, 2020, original scientific article Keywords: neuroinflammation, neurodegeneration, lipopolysaccharide, glia, cathepsin X, neuroprotection Full text (file, 7,62 MB) This document has more files! More... |
67. ATP-competitive inhibitors of human DNA topoisomerase IIα with improved antiproliferative activity based on N-phenylpyrrolamide scaffoldŽiga Skok, Martina Durcik, Živa Zajec, Darja Gramec, Krištof Bozovičar, Anja Pišlar, Tihomir Tomašič, Anamarija Zega, Lucija Peterlin-Mašič, Danijel Kikelj, Nace Zidar, Janez Ilaš, 2023, original scientific article Keywords: anticancer drugs, ATP-competitive inhibitors, catalytic inhibitor, cytotoxicity, human DNA topoisomerase II Full text (file, 2,83 MB) This document has more files! More... |
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70. Sinteza in vrednotenje novih N-(4-karbamoilfenil)pirolamidnih zaviralcev človeške DNA-topoizomeraze IINataša Turk, 2019, master's thesis Keywords: DNA-topoizomeraza II, protirakave učinkovine, ATP-kompetitivni zaviralci, N-(4-karbamoilfenil)pirolamidi, zaviralci angiogeneze, zaviralci sinteze DNA, sinteza spojin, sintezni postopki Full text (file, 1,59 MB) |