31. Selective DNA gyrase inhibitorsTihomir Tomašič, Asta Zubrienė, Žiga Skok, Riccardo Martini, Stane Pajk, Izidor Sosič, Janez Ilaš, Daumantas Matulis, Sharon D. Bryant, 2021, original scientific article Keywords: antibacterial, ATP-competitive, DNA gyrase, Hsp90, pharmacophore model, topoisomerase II, target activity profiling, topoisomerase IIα Full text (file, 6,96 MB) This document has more files! More... |
32. Hybrid inhibitors of DNA gyrase A and BMartina Durcik, Žiga Skok, Janez Ilaš, Nace Zidar, Anamarija Zega, Petra Szili, Gábor Draskovits, T. Revesz, Danijel Kikelj, Ákos Nyerges, Csaba Pál, Lucija Peterlin-Mašič, Tihomir Tomašič, 2021, original scientific article Keywords: antibacterial, ciprofloxacin, DNA gyrase, dual inhibitor, hybrid Full text (file, 3,42 MB) This document has more files! More... |
33. Discovery of benzothiazole scaffold-based DNA gyrase B inhibitorsMarina Gjorgjieva, Tihomir Tomašič, Michaela Barančokova, Sotirios Katsamakas, Janez Ilaš, Päivi Tammela, Lucija Peterlin-Mašič, Danijel Kikelj, 2016, original scientific article Keywords: organoruthenium complexes, diketonates, anticancer drugs, ROS, cytotoxicity, cell cycle arrest Full text (file, 1,17 MB) This document has more files! More... |
|
35. Exploring the chemical space of benzothiazole-based DNA gyrase B inhibitorsŽiga Skok, Michaela Barančokova, Ondřej Benek, Cristina Durante Cruz, Päivi Tammela, Tihomir Tomašič, Nace Zidar, Lucija Peterlin-Mašič, Anamarija Zega, Danijel Kikelj, Janez Ilaš, 2020, original scientific article Keywords: DNA gyrase, topoisomerase IV, GyrB, ParE, antibacterial benzothiazole Full text (file, 2,22 MB) This document has more files! More... |
36. Efficient synthesis of hydroxy-substituted 2-aminobenzo[d]thiazole-6-carboxylic acid derivatives as new building blocks in drug discoveryMartina Durcik, Žan Toplak, Nace Zidar, Janez Ilaš, Anamarija Zega, Danijel Kikelj, Lucija Peterlin-Mašič, Tihomir Tomašič, 2020, original scientific article Keywords: benzo[d]thiazol, medicinal chemistry Full text (file, 1,03 MB) This document has more files! More... |
37. Rational design of balanced dual-targeting antibiotics with limited resistanceÁkos Nyerges, Tihomir Tomašič, Martina Durcik, T. Revesz, Petra Szili, Žiga Skok, Nace Zidar, Janez Ilaš, Anamarija Zega, Danijel Kikelj, Lucija Peterlin-Mašič, 2020, original scientific article Keywords: antibiotics, bacterial resistance, bacterial targets Full text (file, 2,33 MB) This document has more files! More... |
38. Next-generation heterocyclic electrophiles as small-molecule covalent MurA inhibitorsPéter Ábrányi-Balogh, Aaron Keeley, György G. Ferenczy, László Petri, Tímea Imre, Katarina Grabrijan, Martina Hrast, Damijan Knez, Janez Ilaš, Stanislav Gobec, György Keserü M., 2022, original scientific article Keywords: covalent inhibitor, heterocyclic electrophiles, cysteine labelling, quaternization, MurA Full text (file, 1,46 MB) This document has more files! More... |
39. Discovery and hit-to-lead optimization of benzothiazole scaffold-based DNA gyrase inhibitors with potent activity against Acinetobacter baumannii and Pseudomonas aeruginosaAndrej Emanuel Cotman, Martina Durcik, Davide Benedetto Tiz, Federica Fulgheri, Daniela Secci, Maša Sterle, Štefan Možina, Žiga Skok, Nace Zidar, Anamarija Zega, Janez Ilaš, Lucija Peterlin-Mašič, Tihomir Tomašič, Danijel Kikelj, 2023, original scientific article Keywords: antibacterial activity, bacteria, genetics, inhibitors, solubility Full text (file, 7,98 MB) This document has more files! More... |
40. Exploring the 5-substituted 2-aminobenzothiazole-based DNA gyrase B inhibitors active against ESKAPE pathogensMaša Sterle, Martina Durcik, Danijel Kikelj, Nace Zidar, Lucija Peterlin-Mašič, Janez Ilaš, Tihomir Tomašič, Andrej Emanuel Cotman, Anamarija Zega, 2023, original scientific article Keywords: bacteria, genetics, inhibitors, organic acids, peptides, proteins Full text (file, 4,52 MB) This document has more files! More... |