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1. Design and synthesis of novel 3-triazolyl-1-thiogalactosides as galectin-1, -3 and -8 inhibitors Sjors van Klaveren, Jaka Dernovšek, Žiga Jakopin, Marko Anderluh, Hakon Leffler, Ulf Nilsson, Tihomir Tomašič, 2022, izvirni znanstveni članek Celotno besedilo (datoteka, 1010,75 KB) Gradivo ima več datotek! Več... |
2. Small-Molecule Galectin Ligands: Structure-Based Optimisation of Affinity and Selectivity Sjors Van Klaveren, 2024, doktorsko delo/naloga Ključne besede: Galectins, ligands, inhibitors, drug discovery, molecular dynamics simulations, virtual screening, docking studies, structure-activity relationship, X-ray crystallography. |