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1. Discovery of substituted oxadiazoles as a novel scaffold for DNA gyrase inhibitors Žiga Jakopin, Janez Ilaš, Michaela Barančokova, Matjaž Brvar, Päivi Tammela, Marija Sollner Dolenc, Tihomir Tomašič, Danijel Kikelj, 2017, original scientific article Keywords: 1, 2, 4-oxadiazoles, DNA gyrase inhibition, topoisomerase IV inhibition, antibacterial screening, computer-aided drug design |
2. Design and synthesis of 3,5-substituted 1,2,4-oxadiazoles as catalytic inhibitors of human DNA topoisomerase ▫$II\alpha$▫ Kaja Bergant Loboda, Katja Valjavec, Martina Štampar, Gerhard Wolber, Bojana Žegura, Metka Filipič, Marija Sollner Dolenc, Andrej Perdih, 2020, original scientific article Keywords: human DNA topoisomerase II[alpha], catalytic inhibitors, drug design, oxadiazoles, anticancer agents |