1. Synthesis, molecular modelling and biological evaluation of novel heterodimeric, multiple ligands targeting cholinesterases and amyloid betaMichalina Hebda, Marek Bajda, Anna Więckowska, Natalia Szałaj, Anna Pasieka, Dawid Panek, Justyna Godyń, Tomasz Wichur, Damijan Knez, Stanislav Gobec, Barbara Malawska, 2016, original scientific article Keywords: cholinesterase inhibitors, molecular modelling, β-amyloid aggregation inhibitors, Alzheimer’s disease, multi-target-directed ligands (MTDL), PAMPA-BBB assay
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2. Synthesis and biological evaluation of benzochromenopyrimidinones as cholinesterase inhibitors and potent antioxidant, non-hepatotoxic agents for Alzheimer's diseaseYoussef Dgachi, Oscar M. Bautista-Aguilera, Mohamed Benchekroun, Hélène Martin, Alexandre Bonet, Damijan Knez, Justyna Godyń, Barbara Malawska, Stanislav Gobec, Mourad Chioua, Jana Janockova, Ondrej Soukup, Fakher Chabchoub, José Marco-Contelles, Lhassane Ismaili, 2016, original scientific article Keywords: Alzheimer's disease, quinazolinones, multicomponent reactions, multitarget-directed ligands, antioxidants, cholinesterase inhibitors, hepatotoxicity
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3. Design, synthesis, and biological evaluation of 2-(benzylamino-2-hydroxyalkyl)isoindoline-1,3-diones derivatives as potential disease-modifying multifunctional anti-Alzheimer agentsDawid Panek, Anna Więckowska, Anna Pasieka, Justyna Godyń, Jakub Jończyk, Marek Bajda, Damijan Knez, Stanislav Gobec, Barbara Malawska, 2018, original scientific article Keywords: isoindoline-1, 3-dione derivatives, cholinesterase inhibitors, BACE-1 inhibitors, Aβ-aggregation, molecular modeling, multiple anti-Alzheimer's ligands
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4. From tryptophan-based amides to tertiary aminesAnže Meden, Damijan Knez, Xavier Brazzolotto, Florian Nachon, Jose Dias, Jurij Svete, Jure Stojan, Uroš Grošelj, Stanislav Gobec, 2022, original scientific article Keywords: cholinesterase inhibitors, Alzheimer's disease, butyrylcholinesterase, carbamate, pseudoirreversible inhibition
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5. Spatial distribution and stability of cholinesterase inhibitory protoberberine alkaloids from Papaver setiferumNeda Safa, Tomaž Trobec, Darren C. Holland, Blazej Slazak, Erik Jacobsson, Jeffrey A. Hawkes, Robert Frangež, Kristina Sepčić, Ulf Göransson, Lindon W. K. Moodie, Luke P. Robertson, 2022, original scientific article Keywords: Cholinesterase Inhibitors, Papaver, Alkaloids
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6. Development of potent cholinesterase inhibitors based on a marine pharmacophoreVijayaragavan Elumalai, Tomaž Trobec, Maja Grundner, Christophe Labriere, Robert Frangež, Kristina Sepčić, Jørn H. Hansen, Johan Svenson, 2022, original scientific article Keywords: Nervous System Diseases, Cholinesterase Inhibitors
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7. Potential revival of cholinesterase inhibitors as drugs in veterinary medicineNeža Žnidaršič, Malan Štrbenc, Neža Grgurevič, Tomaž Snoj, 2023, review article Keywords: cholinergic system, cholinesterase inhibitors, organophosphates, carbamates, canine cognitive dysfunction, cognitive dysfunction, dogs
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8. Synthesis and cholinesterase inhibitory activity of selected indole-based compoundsMarija Gršič, Anže Meden, Damijan Knez, Marko Jukič, Jurij Svete, Stanislav Gobec, Uroš Grošelj, 2023, original scientific article Keywords: indole derivatives, tryptophan derivatives, amidations, cholinesterase (ChE) inhibitors, 1, 1’-Carbonyldiimidazole (CDI), rearrangements, catalytic hydrogenation
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