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1. Načrtovanje in sinteza dipeptidnih zaviralcev imunoproteasoma
Katarina Grabrijan, 2017, master's thesis

Keywords: ubikvitin, imunoproteasom, beta5i-podenota, dipeptidni zaviralci, 1, 3, 4-oksatiazol-2-on, psihotropna zdravila
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2. Synthesis of 3-amino-4-substituted monocyclic ß-lactams—important structural motifs in medicinal chemistry
Katarina Grabrijan, Nika Strašek Benedik, Stanislav Gobec, 2022, original scientific article

Keywords: monocyclic ß-lactam, Staudinger [2+2] cyclocondensation, cerium ammonium nitrate, hydrazine hydrate, 3-amino-4-substituted azetidin-2-one, inhibitory activities
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3. Covalent inhibitors of bacterial peptidoglycan biosynthesis enzyme MurA with chloroacetamide warhead
Katarina Grabrijan, Martina Hrast, Matic Proj, Ana Dolšak, Irena Zdovc, Tímea Imre, László Petri, Péter Ábrányi-Balogh, György Keserü M., Stanislav Gobec, 2022, original scientific article

Keywords: antibacterial agents, UDP-N-acetylglucosamine enolpyruvyl transferase, thiol reactivity
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4. Next-generation heterocyclic electrophiles as small-molecule covalent MurA inhibitors
Péter Ábrányi-Balogh, Aaron Keeley, György G. Ferenczy, László Petri, Tímea Imre, Katarina Grabrijan, Martina Hrast, Damijan Knez, Janez Ilaš, Stanislav Gobec, György Keserü M., 2022, original scientific article

Keywords: covalent inhibitor, heterocyclic electrophiles, cysteine labelling, quaternization, MurA
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5. Fragment-sized thiazoles in fragment-based drug discovery campaigns
Matic Proj, Martina Hrast, Damijan Knez, Krištof Bozovičar, Katarina Grabrijan, Anže Meden, Stanislav Gobec, Rok Frlan, 2022, original scientific article

Keywords: thiazoles, hit profiling, promiscuous compounds, frequent hitters, privileged scaffolds, fragments
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6. Synthesis and biochemical evaluation of new 3-amido-4-substituted monocyclic ß-lactams as inhibitors of penicillin-binding protein(s)
Katarina Grabrijan, Nika Strašek Benedik, Alen Krajnc, Krištof Bozovičar, Damijan Knez, Matic Proj, Irena Zdovc, Izidor Sosič, Martina Hrast, Stanislav Gobec, 2024, original scientific article

Keywords: antibacterial agents, monocyclic-β-lactams, penicillin-binding proteins, covalent inhibitors, transpeptidase
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7. Načrtovanje, sinteza in vrednotenje novih kovalentnih zaviralcev encimov MurA in penicilin vezočih proteinov
Katarina Grabrijan, 2023, doctoral dissertation

Keywords: penicilin vezoči proteini, MurA, kovalentni zaviralci, monociklični β-laktami, kloracetamidi
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