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12. Discovery of substituted oxadiazoles as a novel scaffold for DNA gyrase inhibitorsŽiga Jakopin, Janez Ilaš, Michaela Barančokova, Matjaž Brvar, Päivi Tammela, Marija Sollner Dolenc, Tihomir Tomašič, Danijel Kikelj, 2017, original scientific article Keywords: 1, 2, 4-oxadiazoles, DNA gyrase inhibition, topoisomerase IV inhibition, antibacterial screening, computer-aided drug design Full text (file, 1,45 MB) This document has more files! More... |
13. Synthesis and evaluation of N-phenylpyrrolamides as DNA gyrase B inhibitorsMartina Durcik, Päivi Tammela, Michaela Barančokova, Tihomir Tomašič, Janez Ilaš, Danijel Kikelj, Nace Zidar, 2018, original scientific article Keywords: DNA gyrase, GyrB, antibacterials, inhibitors, pyrrolamides Full text (file, 452,68 KB) This document has more files! More... |
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15. New dual inhibitors of bacterial topoisomerases with broad-spectrum antibacterial activity and in vivo efficacy against vancomycin-intermediate Staphylococcus aureusMartina Durcik, Andrej Emanuel Cotman, Žan Toplak, Štefan Možina, Žiga Skok, Maria Vittoria Piras, Nace Zidar, Janez Ilaš, Anamarija Zega, Jurij Trontelj, Danijel Kikelj, Tihomir Tomašič, Lucija Peterlin-Mašič, 2023, original scientific article Keywords: antibacterial activity, bacteria, inhibitors, genetics, inhibition, peptides and proteins Full text (file, 4,53 MB) This document has more files! More... |
16. Načrtovanje, sinteza in vrednotenje novih ATP-kompetitivnih zaviralcev človeške DNA-topoiomeraze II kot potencialnih protirakavih učinkovinŽiga Skok, 2020, doctoral dissertation Keywords: DNA-topoizomeraza II, protirakave učinkovine, funkcija topoizmeraz, testiranje zaviralne aktivnosti, sinteza zaviralcev, sintezni postopki Full text (file, 6,60 MB) |
17. Immunosuppressive effects of new thiophene-based K$_V$1.3 inhibitorsŠpela Gubič, Janez Ilaš, Tihomir Tomašič, Annarosa Arcangeli, Lucija Peterlin-Mašič, 2023, original scientific article Keywords: ion channel, K$_V$1.3 inhibitor, T-lymphocyte, immunosuppressive Full text (file, 2,73 MB) This document has more files! More... |
18. ATP-competitive inhibitors of human DNA topoisomerase IIα with improved antiproliferative activity based on N-phenylpyrrolamide scaffoldŽiga Skok, Martina Durcik, Živa Zajec, Darja Gramec, Krištof Bozovičar, Anja Pišlar, Tihomir Tomašič, Anamarija Zega, Lucija Peterlin-Mašič, Danijel Kikelj, Nace Zidar, Janez Ilaš, 2023, original scientific article Keywords: anticancer drugs, ATP-competitive inhibitors, catalytic inhibitor, cytotoxicity, human DNA topoisomerase II Full text (file, 2,83 MB) This document has more files! More... |
19. Načrtovanje in sinteza gradnikov novih inhibitorjev faktorja XaUroš Trstenjak, 2009, undergraduate thesis Keywords: faktor Xa, rivaroksban, inhibitorji faktorja Xa, metilni estri, sinteza, metode, etilni estri, sinteza, koagulacijska kaskada Full text (outside link) |
20. Sinteza derivatov benzo[b][1,4]dioksina in benzo[b][1,4]oksazina kot gradnikov dualnih antitrombotičnih učinkovinSaša Ciglič, 2011, undergraduate thesis Keywords: antitrombotične učinkovine, tromboza, hemostaza, benzoksazinski derivati, sinteza 2-(metilamino) fenola, sinteza prekurzorjev enantiomerov, sinteza benzo[b][1, 4]oksazinov Full text (outside link) |