51. Crystal structure of RahU, an aegerolysin protein from the human pathogen Pseudomonas aeruginosa, and its interaction with membrane ceramide phosphorylethanolamineEva Kočar, Tea Lenarčič, Vesna Hodnik, Anastasija Panevska, Yunjie Huang, Gregor Bajc, Rok Kostanjšek, Anjaparavanda P. Naren, Peter Maček, Gregor Anderluh, Kristina Sepčić, Marjetka Podobnik, Matej Butala, 2021, original scientific article Keywords: aegerolysins, crystal structure of RahU, ceramide phosphorylethanolamine, biochemistry, lipids, membrane lipids, membrane proteins, microbiology, proteins, sphingolipids, structural biology, X-ray crystallography Full text (file, 2,95 MB) This document has more files! More... |
52. Potent DNA gyrase inhibitors bind asymmetrically to their target using symmetrical bifurcated halogen bondsAnja Kolarič, Thomas Germe, Martina Hrast, Clare E. M. Stevenson, David M. Lawson, Nicolas P. Burton, Judit Vörös, Anthony Maxwell, Nikola Minovski, Marko Anderluh, 2021, original scientific article Keywords: antibacterials, DNA gyrase inhibitors, drug discovery, Staphylococcus aureus, intercalators, novel bacterial topoisomerase inhibitors, NBTIs, symmetrical bifurcated halogen bonds, crystal structure, novel NBTIs mechanism of action, antimicrobials, DNA-binding proteins, drug development, X-ray crystallography Full text (file, 2,00 MB) This document has more files! More... |
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54. New dual inhibitors of bacterial topoisomerases with broad-spectrum antibacterial activity and in vivo efficacy against vancomycin-intermediate Staphylococcus aureusMartina Durcik, Andrej Emanuel Cotman, Žan Toplak, Štefan Možina, Žiga Skok, Maria Vittoria Piras, Nace Zidar, Janez Ilaš, Anamarija Zega, Jurij Trontelj, Danijel Kikelj, Tihomir Tomašič, Lucija Peterlin-Mašič, 2023, original scientific article Keywords: antibacterial activity, bacteria, inhibitors, genetics, inhibition, peptides and proteins Full text (file, 4,53 MB) This document has more files! More... |
55. Intra-species variations of bioactive compounds of two dictyota species from the Adriatic SeaAna Martić, Lara Čižmek, Nikolai Ul'yanovskii, Tina Paradžik, Lucija Perković, Gabrijela Matijević, Tamara Vujović, Marija Baković, Sanja Babić, Dmitry Kosyakov, Polonca Trebše, Rozelindra Čož-Rakovac, 2023, original scientific article Keywords: Dictyota dichotoma, Dictyota fasciola, brown seaweeds, chromatography, toxicity, proteins, carbohydrates, amino acids, bioactivity Full text (file, 2,86 MB) This document has more files! More... |
56. Heterobifunctional ligase recruiters enable pan-degradation of inhibitor of apoptosis proteinsYuen Lam Dora Ng, Aleša Bricelj, Jacqueline A. Jansen, Arunima Murgai, Kirsten Peter, Katherine A. Donovan, Michael Gütschow, Jan Krönke, Christian Steinebach, Izidor Sosič, 2023, original scientific article Keywords: antagonists, degradation, ligands, mixtures, peptides, proteins, pharmaceutical chemistry Full text (file, 5,93 MB) This document has more files! More... |
57. Rapid, direct, noninvasive method to determine the amount of immobilized proteinRok Ambrožič, Rok Mravljak, Aleš Podgornik, 2023, original scientific article Keywords: immobilization, pH transition, protein quantity, monomers, peptides, proteins, theoretical chemistry, computational chemistry, pH Full text (file, 4,73 MB) This document has more files! More... |
58. All-atom simulations reveal the intricacies of signal transduction upon binding of the HLA-E ligand to the transmembrane inhibitory CD94/NKG2A receptorMartin Ljubič, Eva Prašnikar, Andrej Perdih, Jure Borišek, 2023, original scientific article Keywords: cells, ligands, membranes, peptides, proteins, receptors Full text (file, 6,74 MB) This document has more files! More... |
59. Analyte-driven clustering of bio-conjugated magnetic nanoparticlesTilen Potisk, Jurij Sablić, Daniel Svenšek, Elena Sanz-de Diego, Francisco J. Teran, Matej Praprotnik, 2023, original scientific article Keywords: biochemistry, nanoparticles, magnetic nanoparticles, proteins, biosensors, clustering, magnetic dynamics, mesoscopic simulation, nanomedicine Full text (file, 3,42 MB) This document has more files! More... |
60. Tunable heteroaromatic nitriles for selective bioorthogonal click reaction with cysteineMatic Proj, Nika Strašek Benedik, Stane Pajk, Damijan Knez, Izidor Sosič, 2023, original scientific article Keywords: labeling, monomers, nitrogen compounds, peptides, reactivity, proteins Full text (file, 4,39 MB) This document has more files! More... |