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1. Design and synthesis of novel 3-triazolyl-1-thiogalactosides as galectin-1, -3 and -8 inhibitors Sjors van Klaveren, Jaka Dernovšek, Žiga Jakopin, Marko Anderluh, Hakon Leffler, Ulf Nilsson, Tihomir Tomašič, 2022, izvirni znanstveni članek Celotno besedilo (datoteka, 1010,75 KB) Gradivo ima več datotek! Več... |
2. Structure-guided design of D-galactal derivatives with high affinity and selectivity for the galectin-8 n-terminal domain Mujtaba Hassan, Floriane Baussière, Samo Guzelj, Anders Sundin, Maria Håkansson, Rebeka Kovačič, Hakon Leffler, Tihomir Tomašič, Marko Anderluh, Žiga Jakopin, 2021, izvirni znanstveni članek Ključne besede: Galectin-8N, d-galactal, benzimidazole, selectivity, X-ray crystallography, cytokine secretion |